{"id":203,"date":"2021-11-24T11:14:40","date_gmt":"2021-11-24T02:14:40","guid":{"rendered":"http:\/\/achem.okayama-u.ac.jp\/bioorgchem\/WordPress\/?page_id=203"},"modified":"2026-03-25T20:57:47","modified_gmt":"2026-03-25T11:57:47","slug":"presentation","status":"publish","type":"page","link":"http:\/\/achem.okayama-u.ac.jp\/bioorgchem\/presentation","title":{"rendered":"Presentation"},"content":{"rendered":"\n<p style=\"font-size:20px\"><strong>2025\u5e74\u5ea6<\/strong><\/p>\n\n\n\n<p>8.\u300c\u74b0\u5883\u5fdc\u7b54\u578b\u30ea\u30ac\u30f3\u30c9\u3092\u6307\u5411\u3057\u305f\u30dc\u30ed\u30f3\u9178\u2015\u30b9\u30c6\u30ed\u30a4\u30c9\u878d\u5408\u5206\u5b50\u306e\u5408\u6210\u7814\u7a76\u300d<br>\u25cb\u6e05\u6c34 \u8f1d\u7965\u3001\u68da\u5009 \u6df3\u6717\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c106\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2026\u5e743\u670819\u65e5\uff0c[F]1232-3am-03<\/p>\n\n\n\n<p>7.\u300c\u5149\u6d3b\u6027\u5316\u30d1\u30e9\u30b8\u30a6\u30e0\u3092\u89e6\u5a92\u3068\u3059\u308b\u30d3\u30cb\u30eb\u30dc\u30ed\u30f3\u9178\u30a8\u30b9\u30c6\u30eb\u306e\u30e9\u30b8\u30ab\u30eb\u74b0\u5316\u53cd\u5fdc\u306b\u304a\u3051\u308b\u7acb\u4f53\u9078\u629e\u6027\u306e\u5236\u5fa1\u300d<br>\u25cb\u6e9d\u53e3 \u7384\u6a39\u3001\u798f\u57a3\u5185 \u5c2d\u826f\u3001\u5742\u5009 \u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c106\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2026\u5e743\u670819\u65e5\uff0c[F]1232-3am-04<\/p>\n\n\n\n<p>6.\u300c\u03b2,\u03b2-\u30b8\u30dc\u30ea\u30eb\u30a2\u30e9\u30cb\u30f3\u3092\u69cb\u6210\u8981\u7d20\u3068\u3059\u308b\u30da\u30d7\u30c1\u30c9\u56fa\u76f8\u5408\u6210\u300d<br>\u25cb\u65b0\u7530 \u76f4\u4e4b\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c106\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2026\u5e743\u670819\u65e5\uff0c[F]1232-3am-05<\/p>\n\n\n\n<p>5.\u300cDevelopment of the Diels-Alder Reaction of Vinyl Cyclic Allene\u300d<br>Haruki Mizoguchi, Takumi Obata, Taiki Hirai, Manaka Komatsu, Akira Sakakura<br>ISOR-16\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2025\u5e7411\u670821\u65e5\uff0cP-23<\/p>\n\n\n\n<p>4.\u300cSolid-phase Synthesis&nbsp;of \u03b2,\u03b2-diborylalanine-incorporated peptides\u300d<br>Naoyuki Nitta, Haruki Mizoguchi, Akira Sakakura<br>ISOR-16\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2025\u5e7411\u670821\u65e5\uff0cP-23<\/p>\n\n\n\n<p>3.\u300cSynthetic study toward&nbsp;boron-doped&nbsp;steroids, the&nbsp;cyclic boronic acid&nbsp;containing&nbsp;environment-responsive&nbsp;small&nbsp;molecule&nbsp;ligands\u300d<br>Atsuro Tanakura,&nbsp;Teruyoshi Shimizu, Haruki Mizoguchi, and Akira Sakakura<br>ISOR-16\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2025\u5e7411\u670821\u65e5\uff0cP-3<\/p>\n\n\n\n<p>2.\u300c\u30db\u30a6\u7d20\u30a2\u30fc\u30c8\u932f\u4f53\u3068\u6b6a\u307f\u03c0\u7d50\u5408\u306b\u3088\u308b\u5206\u5b50\u69cb\u7bc9\u300d<br>\u6e9d\u53e3 \u7384\u6a39<br>\u7b2c41\u56de\u6709\u6a5f\u5408\u6210\u5316\u5b66\u30bb\u30df\u30ca\u30fc\uff0c\u53d7\u8cde\u8b1b\u6f14\uff0c\u90e1\u5c71\u5e02\u4e2d\u592e\u516c\u6c11\u9928\uff0c2025\u5e749\u670825\u65e5\uff0cA-5<\/p>\n\n\n\n<p>1.\u300c\u30c6\u30eb\u30da\u30ce\u30a4\u30c9\u578b\u591a\u74b0\u6027\u9aa8\u683c\u306e\u52b9\u7387\u7684\u69cb\u7bc9\u3092\u6307\u5411\u3057\u305f\u30d3\u30cb\u30eb\u5316\u74b0\u72b6\u30a2\u30ec\u30f3Diels-Alder\u53cd\u5fdc\u306e\u958b\u767a\u300d<br>\u6e9d\u53e3 \u7384\u6a39\u3001\u5c0f\u5e61 \u5320\u3001\u5e73\u4e95 \u5927\u8cb4\u3001\u5c0f\u677e \u4e07\u83dc\u4f73\u3001\u5742\u5009 \u5f70<br>\u7b2c67\u56de\u5929\u7136\u6709\u6a5f\u5316\u5408\u7269\u8a0e\u8ad6\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u6771\u5317\u5927\u5b66\u6cb3\u5185\u5317\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2025\u5e749\u67089\u65e5\uff0cP1-22<\/p>\n\n\n\n<p><\/p>\n\n\n\n<p style=\"font-size:20px\"><strong>2024\u5e74\u5ea6<\/strong><\/p>\n\n\n\n<p>14.\u300c\u5149\u6d3b\u6027\u5316\u30d1\u30e9\u30b8\u30a6\u30e0\u3092\u7528\u3044\u308b\u30e9\u30b8\u30ab\u30eb\u4ed8\u52a0\uff0d\u74b0\u5316\u30ab\u30b9\u30b1\u30fc\u30c9\u53cd\u5fdc\u306b\u3088\u308b\u74b0\u5f0f\u30dc\u30ed\u30f3\u9178\u30a8\u30b9\u30c6\u30eb\u5408\u6210\u306b\u304a\u3051\u308b\u4e00\u822c\u6027\u306e\u8abf\u67fb\u300d<br>\u798f\u57a3\u5185 \u5c2d\u826f\u3001\u6c60\u2f65 \u9065\u2fb9\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c105\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u95a2\u897f\u5927\u5b66\u5343\u91cc\u5c71\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2025\u5e743\u670827\u65e5\uff0c[F]2403-2am-12<\/p>\n\n\n\n<p>13.\u300c\u03b2,\u03b2-\u30b8\u30dc\u30ea\u30eb\u30a2\u30e9\u30cb\u30f3\u306e\u958b\u767a\u3068\u30da\u30d7\u30c1\u30c9\u5408\u6210\u3078\u306e\u5c55\u958b\u300d<br>\u65b0\u2f65 \u76f4\u4e4b\u3001\u4e2d\u4e95 \u8b19\u2f3c\u3001\u6e9d\u2f1d \u2f5e\u6a39\u3001\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c105\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u95a2\u897f\u5927\u5b66\u5343\u91cc\u5c71\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2025\u5e743\u670827\u65e5\uff0c[F]2403-2am-13<\/p>\n\n\n\n<p>12.\u300c\u30b7\u30af\u30ed\u30d7\u30ed\u307a\u30cb\u30eb\u30dc\u30e9\u30fc\u30c8\u306e\u30e1\u30bf\u30ec\u30fc\u30c8\u8ee2\u4f4d\u3092\u5229\u7528\u3059\u308b\u70ad\u7d20\uff17\u54e1\u74b0\u5408\u6210\u306b\u304a\u3051\u308b\u57fa\u8cea\u9069\u7528\u7bc4\u56f2\u306e\u8abf\u67fb\u300d<br>\u6e9d\u53e3 \u7384\u6a39\u3001\u5c0f\u90f7 \u5609\u5f66\u3001\u82b9\u751f \u5c06\u54c9\u3001\u5742\u5009 \u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c105\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u95a2\u897f\u5927\u5b66\u5343\u91cc\u5c71\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2025\u5e743\u670828\u65e5\uff0c[F]2402-3am-08<\/p>\n\n\n\n<p>11.\u300c\u30d3\u30cb\u30eb\u74b0\u72b6\u30a2\u30ec\u30f3\u3092\u9ad8\u6d3b\u6027\u30b8\u30a8\u30f3\u7a2e\u3068\u3057\u3066\u7528\u3044\u308b Diels-Alder \u53cd\u5fdc\u306e\u958b\u767a\u300d<br>\u6e9d\u53e3 \u7384\u6a39\u3001\u5c0f\u5e61 \u5320\u3001\u5e73\u4e95 \u5927\u8cb4\u3001\u5c0f\u677e \u4e07\u83dc\u4f73\u3001\u5742\u5009 \u5f70<br>\u7b2c51\u56de\u6709\u6a5f\u5178\u578b\u5143\u7d20\u5316\u5b66\u8a0e\u8ad6\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u4eac\u90fd\u5927\u5b66\uff0c2024\u5e7412\u67087\u65e5, 3O-16<\/p>\n\n\n\n<p>10.\u300c\u751f\u5408\u6210\u7d4c\u8def\u3092\u6a21\u5023\u3057\u305f\u30b0\u30e9\u30e4\u30ca\u30f3\u30b8\u30c6\u30eb\u30da\u30ce\u30a4\u30c9\u306e\u5408\u6210\u7814\u7a76\u300d<br>\u938c\u2f65 \u82f1\u5bff\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u7b2c66\u56de\u5929\u7136\u6709\u6a5f\u5316\u5408\u7269\u8a0e\u8ad6\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u4eac\u90fd\u5927\u5b66\uff0c2024\u5e749\u67085\u65e5, P2-17<\/p>\n\n\n\n<p>9.\u300c\u74b0\u7e2e\u2f29\u578b\u30e1\u30bf\u30ec\u30fc\u30c8\u8ee2\u4f4d\u306b\u3088\u308b\u30a4\u30f3\u30c0\u30f3\u5408\u6210\u306b\u304a\u3051\u308b\u2f00\u822c\u6027\u306e\u8abf\u67fb\u300d<br>\u53e4\u5c4b \u6d35\u592a\u90ce\u3001\u2f5a\u2f2d \u53cb\u2fa5\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u7b2c12\u56de \u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e7411\u670817\u65e5, 2B-30<\/p>\n\n\n\n<p>8.\u300c\u2f63\u5408\u6210\u7d4c\u8def\u3092\u6a21\u5023\u3057\u305f\u2fbb\u683c\u8ee2\u4f4d\u3092\u9375\u3068\u3059\u308b grayanane diterpenoid \u306e\u5408\u6210\u7814\u7a76\u300d<br>\u938c\u2f65 \u82f1\u5bff\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u7b2c12\u56de \u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e7411\u670817\u65e5, 2B-28<\/p>\n\n\n\n<p>7.\u300c\u6838\u9593\u4f4d\u8131\u70ad\u9178 Giese \u53cd\u5fdc\u3092\u9375\u3068\u3059\u308b\u30c8\u30ea\u30ad\u30ca\u30f3\u2fbb\u683c\u5408\u6210\u300d<br>\u2ec4\u2f95 \u62d3\u5922\u3001\u677e\u4e38 \u76f4\u7766\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u7b2c12\u56de \u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e7411\u670817\u65e5, 2B-27<\/p>\n\n\n\n<p>6.\u300c\u30d3\u30b9\uff08\u30dc\u30ea\u30f3\u9178\uff09\u89e6\u5a92\u3092\u2f64\u3044\u305f\u30a2\u30df\u30c9\u7e2e\u5408\u53cd\u5fdc\u306e\u958b\u767a\u300d<br>\u6cb3\u91ce \u771f\u5922\u3001\u6d25\u2f65 \u83dc\u3005\u2fb9\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u7b2c12\u56de \u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e7411\u670817\u65e5, 2B-24<\/p>\n\n\n\n<p>5.\u300c\u30d3\u30cb\u30eb\u74b0\u72b6\u30a2\u30ec\u30f3\u3092\u2f64\u3044\u305f Diels-Alder \u53cd\u5fdc\u306e\u958b\u767a\u300d<br>\u5e73\u4e95 \u2f24\u8cb4\u3001\u2f29\u5e61 \u5320\u3001\u2f29\u677e \u4e07\u83dc\u4f73\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u7b2c12\u56de \u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e7411\u670817\u65e5, 2B-24<\/p>\n\n\n\n<p>4.\u300c\u03b1-\u30b1\u30c8\u30a8\u30b9\u30c6\u30eb\u306e\u76f4\u622a\u7684\u4e0d\u2eeb Mannich \u53cd\u5fdc\u306b\u304a\u3051\u308b\u57fa\u8cea\u9069\u2f64\u7bc4\u56f2\u306e\u62e1\u5f35\u306e\u691c\u8a0e\u300d<br>\u2ec4\u2f2d \u667a\u7a00\u3001\u6d25\u2f65 \u83dc\u3005\u2fb9\u3001\u5b89\u90e8 \u5cb3\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u7b2c12\u56de \u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e7411\u670816\u65e5, 1PB-37<\/p>\n\n\n\n<p>3.\u300c\u89e6\u5a92\u7684\u30e9\u30b8\u30ab\u30eb\u4ed8\u52a0\uff0d\u74b0\u5316\u30ab\u30b9\u30b1\u30fc\u30c9\u53cd\u5fdc\u306b\u3088\u308b\u30db\u30a6\u7d20\u7f6e\u63db\uff15\u54e1\u74b0\u69cb\u9020\u306e\u5408\u6210\u300d<br>\u798f\u57a3\u5185 \u5c2d\u826f\u3001\u6c60\u2f65 \u9065\u2fb9\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u7b2c12\u56de \u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e7411\u670816\u65e5, 1PB-36<\/p>\n\n\n\n<p>2.\u300c\u65b0\u898f\u30a2\u30df\u30ce\u9178\u3067\u3042\u308b \u03b2,\u03b2-\u30b8\u30dc\u30ea\u30eb\u30a2\u30e9\u30cb\u30f3\u306e\u958b\u767a\u300d<br>\u65b0\u2f65 \u76f4\u4e4b\u3001\u4e2d\u4e95 \u8b19\u2f3c\u3001\u6e9d\u2f1d \u2f5e\u6a39\u3001\u5742\u5009\u5f70<br>\u7b2c12\u56de \u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e7411\u670816\u65e5, 1PB-22<\/p>\n\n\n\n<p>1.\u300c\u30b1\u30c6\u30f3\u3068\u30d3\u30cb\u30eb\u30dc\u30ed\u30f3\u9178\u30a8\u30b9\u30c6\u30eb\u3068\u306e\u30e1\u30bf\u30ec\u30fc\u30c8\u8ee2\u4f4d\u3092\u4f34\u3046\u30ab\u30c3\u30d7\u30ea\u30f3\u30b0\u53cd\u5fdc\u306e\u958b\u767a\u300d<br>\u68da\u5009 \u6df3\u6717\u3001\u53e4\u89d2 \u840c\u9999\u3001\u7f8e\u5d0e \u66a2\u5b50\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u7b2c12\u56de \u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e7411\u670816\u65e5, 1PB-16<\/p>\n\n\n\n<p style=\"font-size:20px\"><strong>2023\u5e74\u5ea6<\/strong><\/p>\n\n\n\n<p>10.\u300c\u30b1\u30c6\u30f3\u3068\u30d3\u30cb\u30eb\u30dc\u30ed\u30f3\u9178\u30a8\u30b9\u30c6\u30eb\u3068\u306e\u30e1\u30bf\u30ec\u30fc\u30c8\u8ee2\u4f4d\u3092\u4f34\u3046\u30ab\u30c3\u30d7\u30ea\u30f3\u30b0\u306b\u304a\u3051\u308b\u4e00\u822c\u6027\u306e\u8abf\u67fb\u300d<br>\u68da\u5009 \u6df3\u6717\u3001\u53e4\u89d2 \u840c\u9999\u3001\u7f8e\u5d0e \u66a2\u5b50\u3001\u5c0f\u6a4b \u53cb\u54c9\u3001\u5742\u6771 \u660c\u8d77\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c104\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e743\u670818\u65e5\uff0cE1143-1am-04<\/p>\n\n\n\n<p>9.\u300c5,5\u2019\u4f4d\u306b\u30eb\u30a4\u30b9\u5869\u57fa\u6027\u7f6e\u63db\u57fa\u3092\u6709\u3059\u308b\u30ad\u30e9\u30eb\u30d3\u30b9\uff08\u30aa\u30ad\u30b5\u30be\u30ea\u30f3\uff09\u914d\u4f4d\u5b50\u306e\u8a2d\u8a08\u300d<br>\u897f\u5c71 \u667a\u7a00\u3001\u7e8c\u6728 \u96c4\u5927\u3001\u5b89\u90e8 \u5cb3\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c104\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e743\u670818\u65e5\uff0cE1143-1vn-02<\/p>\n\n\n\n<p>8.\u300c\u74b0\u7e2e\u5c0f\u578b\u30e1\u30bf\u30ec\u30fc\u30c8\u8ee2\u4f4d\u306b\u3088\u308b\u591a\u7f6e\u63db\u30a4\u30f3\u30c0\u30f3\u306e\u7acb\u4f53\u9078\u629e\u7684\u69cb\u7bc9\u300d<br>\u6e9d\u53e3 \u7384\u6a39\u3001\u53e4\u5c4b \u6d35\u592a\u90ce\u3001\u7247\u5c71 \u53cb\u91cc\u3001\u7530\u6751 \u7d14\u4e00\u3001\u5742\u5009 \u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c104\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e743\u670819\u65e5\uff0cE1143-2am-04<\/p>\n\n\n\n<p>7.\u300c\u30a2\u30df\u30c9\u7e2e\u5408\u53cd\u5fdc\u306b\u6709\u52b9\u306a\u30d3\u30b9\uff08\u30dc\u30ea\u30f3\u9178\uff09\u89e6\u5a92\u306e\u8a2d\u8a08\u300d<br>\u6d25\u7530 \u83dc\u3005\u9999\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c104\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e743\u670819\u65e5\uff0cE1143-2am-05<\/p>\n\n\n\n<p>6.\u300c\u5149\u6d3b\u6027\u5316\u30d1\u30e9\u30b8\u30a6\u30e0\u3092\u7528\u3044\u308b\u30e9\u30b8\u30ab\u30eb\u4ed8\u52a0\uff0d\u74b0\u5316\u30ab\u30b9\u30b1\u30fc\u30c9\u53cd\u5fdc\u306b\u3088\u308b\u74b0\u5f0f\u30dc\u30ed\u30f3\u9178\u30a8\u30b9\u30c6\u30eb\u5408\u6210\u6cd5\u300d<br>\u798f\u57a3\u5185 \u5c2d\u826f\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u6c60\u7530 \u9065\u9999\u3001\u5742\u5009 \u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c104\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e743\u670820\u65e5\uff0cE1143-3am-01<\/p>\n\n\n\n<p>5.\u300c\u9aa8\u683c\u8ee2\u4f4d\u3092\u9375\u3068\u3059\u308b\u30b0\u30e9\u30e4\u30ca\u30f3\u30b8\u30c6\u30eb\u30da\u30ce\u30a4\u30c9\u306e\u5408\u6210\u7814\u7a76\u300d<br>\u938c\u7530 \u82f1\u5bff\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c104\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e743\u670819\u65e5\uff0cH933-2am-12<\/p>\n\n\n\n<p>4.\u300c\u30d3\u30cb\u30eb\u74b0\u72b6\u30a2\u30ec\u30f3\u3092\u65b0\u898f\u6b6a\u307f\u30b8\u30a8\u30f3\u3068\u3057\u3066\u7528\u3044\u305fDiels-Alder\u53cd\u5fdc\u306e\u958b\u767a\u3068\u70ad\u7d20\u74b0\u9aa8\u683c\u306e\u69cb\u7bc9\u300d<br>\u5c0f\u5e61 \u5320\u3001\u5e73\u4e95 \u5927\u8cb4\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c104\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e743\u670820\u65e5\uff0cH933-3pm-01<\/p>\n\n\n\n<p>3.\u300c\u591a\u74b0\u6027\u30c6\u30eb\u30da\u30f3\u9aa8\u683c\u69cb\u7bc9\u306e\u305f\u3081\u306e\u6838\u9593\u4f4d\u30e9\u30b8\u30ab\u30eb\u30ab\u30c3\u30d7\u30ea\u30f3\u30b0\u53cd\u5fdc\u306e\u958b\u767a\u300d<br>\u677e\u4e38 \u76f4\u7766\u3001\u6e9d\u53e3 \u7384\u6a39\u3001\u5742\u5009 \u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c104\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2024\u5e743\u670820\u65e5\uff0cH933-3pm-02<\/p>\n\n\n\n<p>2.\u300c\u30db\u30a6\u7d20\u30a2\u30fc\u30c8\u932f\u4f53\u306e\u30e1\u30bf\u30ec\u30fc\u30c8\u8ee2\u4f4d\u3092\u4e2d\u5fc3\u3068\u3059\u308b\u5206\u5b50\u69cb\u7bc9\u300d<br>\u6e9d\u53e3\u7384\u6a39<br>\u7b2c37\u56de\u82e5\u624b\u5316\u5b66\u8005\u306e\u305f\u3081\u306e\u5316\u5b66\u9053\u5834\uff0c\u62db\u5f85\u8b1b\u6f14\uff0c\u5e83\u5cf6\u5e02\u56fd\u969b\u9752\u5e74\u4f1a\u9928\uff0c2023\u5e74\uff19\u6708\uff16\u65e5<\/p>\n\n\n\n<p>1.\u300c\u30db\u30a6\u7d20\u304c\u4e3b\u5f79\u3068\u306a\u308b\u30a2\u30fc\u30c8\u306a\u53cd\u5fdc\u306e\u958b\u767a\u3092\u76ee\u6307\u3057\u3066\u300d<br>\u6e9d\u53e3\u7384\u6a39<br>\u7b2c\uff18\u56de\u6709\u6a5f\u82e5\u624b\u30ef\u30fc\u30af\u30b7\u30e7\u30c3\u30d7\uff0c\u62db\u5f85\u8b1b\u6f14\uff0c\u4eac\u90fd\u5927\u5b66\uff0c2023\u5e7412\u67082\uff10\u65e5<\/p>\n\n\n\n<p style=\"font-size:20px\"><strong>2022\u5e74\u5ea6<\/strong><\/p>\n\n\n\n<p>4.\u300c\u30d3\u30b7\u30af\u30ed[3.2.1]\u30aa\u30af\u30bf\u30f3\u74b0\u542b\u6709\u5929\u7136\u7269\u306e\u53ce\u675f\u7684\u9aa8\u683c\u69cb\u7bc9\u6cd5\u306e\u958b\u767a\u300d<br>\u677e\u4e38\u76f4\u7766\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c103\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6771\u4eac\u7406\u79d1\u5927\u5b66\u91ce\u7530\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2023\u5e743\u670825\u65e5\uff0cD1443-3am-02<\/p>\n\n\n\n<p>3.\u300c\u30b0\u30e9\u30e4\u30ca\u30f3\u30b8\u30c6\u30eb\u30da\u30ce\u30a4\u30c9\u306e\u751f\u5408\u6210\u6a21\u5023\u578b\u5408\u6210\u7814\u7a76\u300d<br>\u938c\u7530\u82f1\u5bff\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c103\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6771\u4eac\u7406\u79d1\u5927\u5b66\u91ce\u7530\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2023\u5e743\u670825\u65e5\uff0cD1443-3am-01<\/p>\n\n\n\n<p>2.\u300c\u30b9\u30eb\u30db\u30f3\u30a2\u30df\u30c9\u57fa\u3092\u6709\u3059\u308b\u30ad\u30e9\u30eb\u30eb\u30a4\u30b9\u9178\u89e6\u5a92\u3092\u7528\u3044\u305f\u03b1\u2013\u30b1\u30c8\u30a8\u30b9\u30c6\u30eb\u306e\u76f4\u63a5\u7684\u4e0d\u6589Mannich\u53cd\u5fdc\u300d<br>\u5b89\u90e8 \u5cb3\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c103\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6771\u4eac\u7406\u79d1\u5927\u5b66\u91ce\u7530\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2023\u5e743\u670824\u65e5\uff0cK705-3am-07<\/p>\n\n\n\n<p>1.\u300c\u30db\u30a6\u7d20\u30a2\u30fc\u30c8\u932f\u4f53\u306e\u30e1\u30bf\u30ec\u30fc\u30c8\u8ee2\u4f4d\u3092\u5229\u7528\u3059\u308b\u5206\u5b50\u69cb\u7bc9\u6cd5\u306e\u958b\u767a\u300d<br>\u6e9d\u53e3\u7384\u6a39<br>2022\u5e74\u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a \u5e83\u5cf6\u5927\u4f1a\uff0c\u62db\u5f85\u516c\u6f14\uff0c\u5e83\u5cf6\uff0c2022\u5e7411\u670813\u65e5<\/p>\n\n\n\n<p style=\"font-size:20px\"><strong>2021\u5e74\u5ea6<\/strong><\/p>\n\n\n\n<p>5.\u300c\u30d3\u30b7\u30af\u30ed[3.2.1]\u30aa\u30af\u30bf\u30f3\u74b0\u3092\u6709\u3059\u308b\u591a\u74b0\u6027\u9aa8\u683c\u306e\u5408\u6210 (Synthesis of polycyclic skeletons including bicyclo[3.2.1]octane ring)\u300d<br>\u938c\u7530\u82f1\u5bff\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c102\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u30aa\u30f3\u30e9\u30a4\u30f3\u958b\u50ac\uff0c2022\u5e743\u670826\u65e5\uff0cB104-4pm-14<\/p>\n\n\n\n<p>4.\u300c\u30b7\u30af\u30ed\u30d7\u30ed\u30da\u30cb\u30eb\u30dc\u30ed\u30f3\u9178\u30a8\u30b9\u30c6\u30eb\u30a2\u30fc\u30c8\u932f\u4f53\u306e1,2-\u30e1\u30bf\u30ec\u30fc\u30c8\u8ee2\u4f4d\u3092\u5229\u7528\u3059\u308b\u4e03\u54e1\u74b0\u69cb\u9020\u306e\u69cb\u7bc9 (Construction of seven-membered carbocycles using 1,2-metallate rearrangement of cyclopropenylboronic ester ate-complex)\u300d<br>\u82b9\u751f\u5c06\u54c9\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c102\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u30aa\u30f3\u30e9\u30a4\u30f3\u958b\u50ac\uff0c2022\u5e743\u670824\u65e5\uff0cK307-2am-05<\/p>\n\n\n\n<p>3.\u300c\u30ad\u30e9\u30eb\u30eb\u30a4\u30b9\u9178\u89e6\u5a92\u3092\u7528\u3044\u305f\u76f4\u622a\u7684\u4e0d\u6589\u30a2\u30eb\u30c9\u30fc\u30eb\u53cd\u5fdc\u306b\u3088\u308b\u03b2-\u30d2\u30c9\u30ed\u30ad\u30b7\u56db\u7d1a\u30a2\u30df\u30ce\u9178\u985e\u306e\u7acb\u4f53\u9078\u629e\u7684\u306a\u5408\u6210 (Asymmetric synthesis of&nbsp;b-hydroxy quaternary amino acids via chiral Lewis acid-catalyzed direct aldol reaction)\u300d<br>\u8352\u6728\u96c4\u4e5f\uff0c\u82b1\u7530\u5c06\u4eba\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c102\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u30aa\u30f3\u30e9\u30a4\u30f3\u958b\u50ac\uff0c2022\u5e743\u670824\u65e5\uff0cK307-2am-06<\/p>\n\n\n\n<p>2.\u300c\u30b1\u30c6\u30f3\u3067\u99c6\u52d5\u3059\u308b\u30d3\u30cb\u30eb\u30dc\u30ed\u30f3\u9178\u30a8\u30b9\u30c6\u30eb\u30a2\u30fc\u30c8\u932f\u4f53\u306e1,2-\u30e1\u30bf\u30ec\u30fc\u30c8\u8ee2\u4f4d\u53cd\u5fdc\u306e\u958b\u767a (Development of a conjunctive cross-coupling of vinylboronic ester ate-complex with ketene)\u300d<br>\u6e9d\u53e3\u7384\u6a39\uff0c\u53e4\u89d2\u840c\u9999\uff0c\u5409\u7530\u7adc\u58eb\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c102\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u30aa\u30f3\u30e9\u30a4\u30f3\u958b\u50ac\uff0c2022\u5e743\u670826\u65e5\uff0cK5-4am-12<\/p>\n\n\n\n<p>1.\u300c\u30db\u30a6\u7d20\u30a2\u30fc\u30c8\u932f\u4f53\u306e1,2-\u30e1\u30bf\u30ec\u30fc\u30c8\u8ee2\u4f4d\u3092\u6d3b\u7528\u3059\u308b\u30ab\u30c3\u30d7\u30ea\u30f3\u30b0\u53cd\u5fdc\u306e\u958b\u767a\u300d<br>\u6e9d\u53e3\u7384\u6a39<br>\u82e5\u624b\u7814\u7a76\u8005\u306e\u305f\u3081\u306e\u6709\u6a5f\u5316\u5b66\u672d\u5e4c\u30bb\u30df\u30ca\u30fc\uff0c\u62db\u5f85\u516c\u6f14\uff0c\u30aa\u30f3\u30e9\u30a4\u30f3\u958b\u50ac\uff0c2021\u5e7411\u670817\u65e5<\/p>\n\n\n\n<p style=\"font-size:20px\"><strong>2020\u5e74\u5ea6<\/strong><\/p>\n\n\n\n<p>7.\u300c\u03b1-\u30b1\u30c8\u30a8\u30b9\u30c6\u30eb\u306e\u76f4\u622a\u7684\u4e0d\u6589Mannich\u53cd\u5fdc\u306b\u6709\u52b9\u306a\u30ad\u30e9\u30eb\u9285(II)\u89e6\u5a92\u306e\u8a2d\u8a08 (Design of Chiral Lewis Acid Catalyst for the Asymmetric Direct Mannich Reaction of \u03b1-Ketoesters)\u300d<br>\u8fd1\u85e4\u771f\u7531\uff0c\u5ca9\u6728\u4f38\u7a4f\uff0c\u4e09\u5b85\u9ebb\u7531\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c101\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u30aa\u30f3\u30e9\u30a4\u30f3\u958b\u50ac\uff0c2021\u5e743\u670819\u65e5\uff0cA20-3am-16<\/p>\n\n\n\n<p>6.\u300c\u30ad\u30e9\u30eb\u6709\u6a5f\u30a2\u30f3\u30e2\u30cb\u30a6\u30e0\u5869\u89e6\u5a92\u3092\u7528\u3044\u305f3-\u30cb\u30c8\u30ed\u30af\u30de\u30ea\u30f3\u306e\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u7684Diels\u2013Alder\u53cd\u5fdc (Enantioselective Diels\u2013Alder Reaction of 3-Nitrocoumarins Promoted by Chiral organoammonium Salt Catalysts)\u300d<br>\u85e4\u7530\u5553\u592a\uff0c\u6749\u539f\u65e9\u7d00\uff0c\u8352\u6728\u96c4\u4e5f\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c101\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u30aa\u30f3\u30e9\u30a4\u30f3\u958b\u50ac\uff0c2021\u5e743\u670819\u65e5\uff0cA20-3am-11<\/p>\n\n\n\n<p>5.\u300c\u5149\u52b1\u8d77\u3057\u305f\u30d1\u30e9\u30b8\u30a6\u30e0\u89e6\u5a92\u306b\u3088\u308b\u30d9\u30f3\u30b8\u30eb\u30a2\u30eb\u30b3\u30fc\u30eb\u8a98\u5c0e\u4f53\u306e\u5206\u5b50\u5185\uff23\uff0d\uff28\u30b7\u30ea\u30eb\u30e1\u30c1\u30eb\u5316\u53cd\u5fdc\u306e\u958b\u767a (Development of an intramolecular C\u2012H silylmethylation of benzyl alcohol derivatives utilizing photoexcited palladium complex)\u300d<br>\u5409\u7530\u7adc\u58eb\uff0c\u6c60\u7530\u9065\u9999\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c101\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u30aa\u30f3\u30e9\u30a4\u30f3\u958b\u50ac\uff0c2021\u5e743\u670819\u65e5\uff0cA21-2am-08<\/p>\n\n\n\n<p>4.\u300c\u30a4\u30f3\u30c9\u30fc\u30eb\u30c6\u30eb\u30da\u30f3\u985e\u306b\u5171\u901a\u3059\u308b\u9023\u7d9a\u4e0d\u6589\u7b2c\u56db\u7d1a\u70ad\u7d20\u306e\u69cb\u7bc9 (Stereoselective Construction of Contiguous Asymmetric Quaternary Carbon Centers of Indole Terpenes)\u300d<br>\u677e\u4e38\u76f4\u7766\uff0c\u5742\u5009\u5f70\uff0c\u65e9\u5ddd\u4e00\u90ce<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c101\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u30aa\u30f3\u30e9\u30a4\u30f3\u958b\u50ac\uff0c2021\u5e743\u670819\u65e5\uff0cA22-2am-05<\/p>\n\n\n\n<p>3.\u300c\u30a2\u30e9\u30a4\u30f3\u3092\u30c8\u30ea\u30ac\u30fc\u3068\u3059\u308b\u30d3\u30cb\u30eb\u30dc\u30ed\u30f3\u9178\u30a8\u30b9\u30c6\u30eb\u30a2\u30fc\u30c8\u932f\u4f53\u306e1,2-\u30e1\u30bf\u30ec\u30fc\u30c8\u8ee2\u4f4d\u306b\u304a\u3051\u308b\u57fa\u8cea\u9069\u7528\u7bc4\u56f2\u304a\u3088\u3073\u53cd\u5fdc\u6a5f\u69cb\u7814\u7a76 (Mechanistic investigation and substrate scope evaluation of an aryne-triggered 1,2-metallate rearrangement of vinylboronic esters)\u300d<br>\u6e9d\u53e3\u7384\u6a39\uff0c\u68ee\u672c\u4e00\u6a39\uff0c\u938c\u7530\u82f1\u5bff\uff0c\u5409\u7530\u7adc\u58eb\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c101\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u30aa\u30f3\u30e9\u30a4\u30f3\u958b\u50ac\uff0c2021\u5e743\u670819\u65e5\uff0cA19-1am-10<\/p>\n\n\n\n<ol start=\"2\" class=\"wp-block-list\">\n<li>\u300c\u30d3\u30cb\u30eb\u30dc\u30ed\u30f3\u9178\u30a8\u30b9\u30c6\u30eb\u30a2\u30fc\u30c8\u932f\u4f53\u3068\u30a2\u30e9\u30a4\u30f3\u3092\u7d44\u307f\u5408\u308f\u305b\u308b\u591a\u7f6e\u63db\u30a2\u30eb\u30ad\u30eb\u30dc\u30ed\u30f3\u9178\u5408\u6210\u6cd5\u306e\u958b\u767a (Synthesis of highly substituted boronic ester utilized aryne-triggered 1,2-metallate rearrangement of vinylboronic ester)\u300d<br>\u938c\u7530\u82f1\u5bff\uff0c\u68ee\u672c\u4e00\u6a39\uff0c\u5409\u7530\u7adc\u4e8c\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c101\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u30aa\u30f3\u30e9\u30a4\u30f3\u958b\u50ac\uff0c2021\u5e743\u670819\u65e5\uff0cA19-1am-09<\/li>\n<\/ol>\n\n\n\n<ol class=\"wp-block-list\">\n<li>\u300c\u30a4\u30f3\u30c9\u30fc\u30eb\u30b8\u30c6\u30eb\u30da\u30f3\u306e\u7db2\u7f85\u7684\u5408\u6210\u7814\u7a76 (Towards the diversity-oriented synthesis of indole diterpenes)\u300d<br>\u677e\u4e38\u76f4\u7766\uff0c\u5742\u5009\u5f70\uff0c\u65e9\u5ddd\u4e00\u90ce<br>\u7b2c62\u56de\u5929\u7136\u6709\u6a5f\u5316\u5408\u7269\u8a0e\u8ad6\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u30aa\u30f3\u30e9\u30a4\u30f3\u958b\u50ac\uff0c2020\u5e749\u670822\u301c24\u65e5\uff0cP2-9<\/li>\n<\/ol>\n\n\n\n<p><\/p>\n\n\n\n<p style=\"font-size:20px\"><strong>2019\u5e74\u5ea6<\/strong><\/p>\n\n\n\n<p>9.\u300c\u30c6\u30eb\u30da\u30f3\u30c9\u30fc\u30ebE\u306e\u9023\u7d9a\u4e0d\u6589\u7b2c\u56db\u7d1a\u70ad\u7d20\u306e\u5408\u6210\u7814\u7a76 (Synthetic Study of Terpendole E: Stereoselective Construction of Contiguous Asymmetric Quaternary Carbon Centers)\u300d<br>\u677e\u4e38\u76f4\u7766\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c100\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6771\u4eac\u7406\u79d1\u5927\u5b66\u91ce\u7530\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2020\u5e743\u670825\u65e5\uff0c4H6-17\uff08COVID-19\u306e\u305f\u3081\u5b66\u4f1a\u4e2d\u6b62\uff0c\u8b1b\u6f14\u4e88\u7a3f\u96c6\u306e\u767a\u884c\u306b\u3088\u308a\u767a\u8868\u6210\u7acb\uff09<\/p>\n\n\n\n<p>8.\u300c\u975e\u5bfe\u79f0\u5316\u3092\u4f34\u3046\u9084\u5143\u7684Heck\u53cd\u5fdc\u306b\u3088\u308b\u9ad8\u9178\u5316\u578b\u30c6\u30eb\u30da\u30ce\u30a4\u30c9\u9aa8\u683c\u306e\u69cb\u7bc9 (Expeditious Construction of Highly Oxygenated Terpenoid Skeletons Utilizing Desymmetrizing Reductive-Heck Cyclization)\u300d<br>\u5409\u7530\u7adc\u58eb\uff0c\u4e45\u4fdd\u8475\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c100\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6771\u4eac\u7406\u79d1\u5927\u5b66\u91ce\u7530\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2020\u5e743\u670823\u65e5\uff0c2H6-50\uff08COVID-19\u306e\u305f\u3081\u5b66\u4f1a\u4e2d\u6b62\uff0c\u8b1b\u6f14\u4e88\u7a3f\u96c6\u306e\u767a\u884c\u306b\u3088\u308a\u767a\u8868\u6210\u7acb\uff09<\/p>\n\n\n\n<p>7.\u300c\u30ad\u30e9\u30eb\u30eb\u30a4\u30b9\u9178\u89e6\u5a92\u3092\u7528\u3044\u305f\u03b1,\u03b1-\u4e8c\u7f6e\u63db-\u03b2-\u30d2\u30c9\u30ed\u30ad\u30b7-\u03b1-\u30a2\u30df\u30ce\u9178\u69cb\u9020\u306e\u7acb\u4f53\u9078\u629e\u7684\u69cb\u7bc9\u6cd5\u306e\u958b\u767a (Investigation of Stereoselective Construction of \u03b1,\u03b1-Disubstituted \u03b2-Hydroxy-\u03b1-Amino Acid Structure Using Chiral Lewis Acid Catalysts)\u300d<br>\u82b1\u7530\u5c06\u4eba\uff0c\u8352\u6728\u96c4\u4e5f\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c100\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6771\u4eac\u7406\u79d1\u5927\u5b66\u91ce\u7530\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2020\u5e743\u670823\u65e5\uff0c2B4-49\uff08COVID-19\u306e\u305f\u3081\u5b66\u4f1a\u4e2d\u6b62\uff0c\u8b1b\u6f14\u4e88\u7a3f\u96c6\u306e\u767a\u884c\u306b\u3088\u308a\u767a\u8868\u6210\u7acb\uff09<\/p>\n\n\n\n<p>6.\u300c\u30a2\u30e9\u30a4\u30f3\u3092\u30c8\u30ea\u30ac\u30fc\u3068\u3059\u308b\u30d3\u30cb\u30eb\u30dc\u30ed\u30f3\u9178\u30a8\u30b9\u30c6\u30eb\u30a2\u30fc\u30c8\u932f\u4f53\u306e\u6b6a\u307f\u958b\u653e\u578b\u30e1\u30bf\u30ec\u30fc\u30c8\u8ee2\u4f4d\u53cd\u5fdc\u306e\u958b\u767a (Development of a Conjunctive-cross Coupling of Alkenylboronic Ester Ate-complex Enabled by an Aryne Triggered Strain-release 1,2-Metallate Rearrangement)\u300d<br>\u6e9d\u53e3\u7384\u6a39\uff0c\u68ee\u672c\u4e00\u6a39\uff0c\u8c4a\u7530\u8015\u5e73\uff0c\u4ef2\u5b97\u6839\u793c\u5b50\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c100\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6771\u4eac\u7406\u79d1\u5927\u5b66\u91ce\u7530\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2020\u5e743\u670822\u65e5\uff0c1B4-53\uff08COVID-19\u306e\u305f\u3081\u5b66\u4f1a\u4e2d\u6b62\uff0c\u8b1b\u6f14\u4e88\u7a3f\u96c6\u306e\u767a\u884c\u306b\u3088\u308a\u767a\u8868\u6210\u7acb\uff09<\/p>\n\n\n\n<p>5.\u300c\u30db\u30a6\u7d20\u30a2\u30fc\u30c8\u932f\u4f53\u306e1,2-\u30e1\u30bf\u30ec\u30fc\u30c8\u8ee2\u4f4d\u3092\u6d3b\u7528\u3059\u308b\u591a\u7f6e\u63db\u30b7\u30af\u30ed\u30d7\u30ed\u30d4\u30eb\u30dc\u30ed\u30f3\u9178\u306e\u7acb\u4f53\u9078\u629e\u7684\u69cb\u7bc9 (Stereoselective construction of highly substituted cyclopropylboronic esters enabled by 1,2-metallate rearrangement of boron-ate complex)\u300d<br>\u82b9\u751f\u5c06\u54c9\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c100\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6771\u4eac\u7406\u79d1\u5927\u5b66\u91ce\u7530\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2020\u5e743\u670822\u65e5\uff0c1B4-52\uff08COVID-19\u306e\u305f\u3081\u5b66\u4f1a\u4e2d\u6b62\uff0c\u8b1b\u6f14\u4e88\u7a3f\u96c6\u306e\u767a\u884c\u306b\u3088\u308a\u767a\u8868\u6210\u7acb\uff09<\/p>\n\n\n\n<p>4.\u300c\u30b7\u30c7\u30ed\u30d5\u30a9\u30a2\u30c8\u30ea\u30da\u30d7\u30c1\u30c9\u3000\u30b3\u30d7\u30ea\u30ce\u30d5\u30a7\u30ea\u30f3\u306e\u5408\u6210\u3068\u751f\u7269\u6d3b\u6027 (Synthesis and Biological Evaluation of Coprinoferrin)\u300d<br>\u7912\u8c37\u667a\u8f1d\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u6052\u677e\u96c4\u592a\uff0c\u9ad8\u897f\u6f64\uff0c\u6d45\u4e95\u3057\u307b\u308a\uff0c\u6e21\u8fba\u8ce2\u4e8c\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c100\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6771\u4eac\u7406\u79d1\u5927\u5b66\u91ce\u7530\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2020\u5e743\u670822\u65e5\uff0c1H6-40\uff08COVID-19\u306e\u305f\u3081\u5b66\u4f1a\u4e2d\u6b62\uff0c\u8b1b\u6f14\u4e88\u7a3f\u96c6\u306e\u767a\u884c\u306b\u3088\u308a\u767a\u8868\u6210\u7acb\uff09<\/p>\n\n\n\n<p>3.\u300c\u30a2\u30eb\u30c6\u30df\u30b7\u30b8\u30f3\u985e\u306e\u30b7\u30af\u30ed\u30da\u30f3\u30bf\u30f3\u90e8\u306e\u7acb\u4f53\u9078\u629e\u7684\u5408\u6210\u7814\u7a76\u300d<br>\u65e9\u5ddd\u4e00\u90ce\uff0c\u6c38\u6613\u674f\u83dc\uff0c\u5742\u5009\u5f70<br>\u7b2c116\u56de\u6709\u6a5f\u5408\u6210\u30b7\u30f3\u30dd\u30b8\u30a6\u30e02019\u3010\u79cb\u3011\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e9\u7a32\u7530\u5927\u5b66\u56fd\u969b\u4f1a\u8b70\u5834\uff0c2019\u5e7411\u67081\u65e5\uff0cO-38<\/p>\n\n\n\n<ol start=\"2\" class=\"wp-block-list\">\n<li>\u300c\u4eba\u3068\u306f\u4e00\u5473\u9055\u3046\u30aa\u30ec\u6d41\u5929\u7136\u7269\u5408\u6210\u300d<br>\u65e9\u5ddd\u4e00\u90ce<br>\u65e5\u672c\u5316\u5b66\u4f1a\u79cb\u5b63\u4e8b\u696d\u3000\u7b2c9\u56deCSJ\u5316\u5b66\u30d5\u30a7\u30b9\u30bf2019\u3000\u30c6\u30fc\u30de\u4f01\u753b\u30b7\u30f3\u30dd\u30b8\u30a6\u30e0\u300e\u3048\uff1f\uff01\u305d\u3053\u306b\u3053\u3060\u308f\u308b\u6709\u6a5f\u5408\u6210\u5316\u5b66\uff1f\u300f\uff0c\u62db\u5f85\u8b1b\u6f14\uff0c\u30bf\u30ef\u30fc\u30db\u30fc\u30eb\u8239\u5800\uff0c2019\u5e7410\u670816\u65e5<\/li>\n<\/ol>\n\n\n\n<ol class=\"wp-block-list\">\n<li>\u300c\u30b8\u30a2\u30b9\u30c6\u30ec\u30aa\u9078\u629e\u7684Henry\u53cd\u5fdc\u3092\u9375\u3068\u3059\u308b\u30de\u30f3\u30b6\u30b7\u30b8\u30f3B\u306e\u5f62\u5f0f\u5168\u5408\u6210\u300d<br>\u8352\u6728\u96c4\u4e5f\uff0c\u4e09\u597d\u590f\u7f8e\uff0c\u68ee\u672c\u4e00\u6a39\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u7b2c61\u56de\u5929\u7136\u6709\u6a5f\u5316\u5408\u7269\u8a0e\u8ad6\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5e83\u5cf6\u56fd\u969b\u4f1a\u8b70\u5834\uff0c2018\u5e749\u670811\u301c13\u65e5\uff0cP1-14<\/li>\n<\/ol>\n\n\n\n<p style=\"font-size:20px\"><strong>2018\u5e74\u5ea6<\/strong><\/p>\n\n\n\n<ol start=\"7\" class=\"wp-block-list\">\n<li>\u300c\u30e6\u30ba\u30ea\u30df\u30f3\u985e\u306e\u8907\u7d20\u74b0\u90e8\u5206\u306e\u7acb\u4f53\u9078\u629e\u7684\u5408\u6210\u7814\u7a76 (Synthetic Study of Yuzurimine-Type Alkaloids: Stereoselective Construction of Heterocyclic Portion)\u300d<br>\u65e9\u5ddd\u4e00\u90ce\uff0c\u9577\u8c37\u4eae\u4ecb\uff0c\u6c60\u7530\u5c06\u898f\uff0c\u5742\u5009 \u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c99\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u7532\u5357\u5927\u5b66\u5ca1\u672c\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2019\u5e743\u670817\u65e5\uff0c2F2-29<\/li>\n<\/ol>\n\n\n\n<ol start=\"6\" class=\"wp-block-list\">\n<li>\u300c\u30a2\u30eb\u30c6\u30df\u30b7\u30b8\u30f3\u985e\u306e\u30b7\u30af\u30ed\u30da\u30f3\u30bf\u30f3\u90e8\u5206\u306e\u7acb\u4f53\u9078\u629e\u7684\u5408\u6210\u7814\u7a76 (Synthetic Studies of Altemicidin-type Alkaloids: Stereoselective Construction of Cyclopentane Portion)\u300d<br>\u6c38\u6613\u674f\u83dc\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c99\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u7532\u5357\u5927\u5b66\u5ca1\u672c\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2019\u5e743\u670817\u65e5\uff0c2F2-28<\/li>\n<\/ol>\n\n\n\n<ol start=\"5\" class=\"wp-block-list\">\n<li>\u300c\u30b8\u30a2\u30b9\u30c6\u30ec\u30aa\u9078\u629e\u7684Henry\u53cd\u5fdc\u3092\u9375\u53cd\u5fdc\u3068\u3059\u308b\u30de\u30f3\u30b6\u30b7\u30b8\u30f3A\u3001B\u304a\u3088\u3073C\u306e\u5408\u6210\u7814\u7a76 (Synthetic study of manzacidins A, B and C based on diastereoselective Henry reaction)\u300d<br>\u8352\u6728\u96c4\u4e5f\uff0c\u4e09\u597d\u590f\u7f8e\uff0c\u68ee\u672c\u4e00\u6a39\uff0c\u5de5\u85e4\u5b5d\u5e78\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c99\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u7532\u5357\u5927\u5b66\u5ca1\u672c\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2019\u5e743\u670817\u65e5\uff0c2F2-05<\/li>\n<\/ol>\n\n\n\n<ol start=\"4\" class=\"wp-block-list\">\n<li>\u300c\u30ad\u30e9\u30eb\u9285(II)\u89e6\u5a92\u3092\u7528\u3044\u305f\u03b1-\u30b1\u30c8\u30a8\u30b9\u30c6\u30eb\u306e\u76f4\u622a\u7684\u306a\u4e0d\u6589Mannich\u53cd\u5fdc\u306e\u958b\u767a (Investigation of Asymmetric Direct Mannich Reaction of \u03b1-Ketoesters Promoted by Chiral Lewis Acid Catalyst)\u300d<br>\u4e09\u5b85\u9ebb\u7531\uff0c\u91cd\u68ee\u572d\u4ecb\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c99\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u7532\u5357\u5927\u5b66\u5ca1\u672c\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2019\u5e743\u670817\u65e5\uff0c2E6-05<\/li>\n<\/ol>\n\n\n\n<ol start=\"3\" class=\"wp-block-list\">\n<li>\u300c\u30ad\u30e9\u30eb\u6709\u6a5f\u30a2\u30f3\u30e2\u30cb\u30a6\u30e0\u5869\u89e6\u5a92\u3092\u7528\u3044\u305f\u30cb\u30c8\u30ed\u30f3\u3068\u03b1-\u7f6e\u63db\u578b\u30a2\u30af\u30ed\u30ec\u30a4\u30f3\u3068\u306e\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u76841,3-\u53cc\u6975\u5b50\u74b0\u5316\u4ed8\u52a0\u53cd\u5fdc (Enantioselective 1,3-Dipolar Cycloaddition of \u03b1-Substituted acroleins with Nitrones Catalyzed by Chiral Organoammonium salts)\u300d<br>\u9b3c\u7ae5\u3061\u3072\u308d\uff0c\u6e9d\u53e3\u7384\u6a39\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c99\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u7532\u5357\u5927\u5b66\u5ca1\u672c\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2019\u5e743\u670817\u65e5\uff0c2E6-04<\/li>\n<\/ol>\n\n\n\n<ol start=\"2\" class=\"wp-block-list\">\n<li>\u300c\u30ad\u30e9\u30eb\u306a\u30d6\u30ec\u30f3\u30b9\u30c6\u30c3\u30c9\u9178\u89e6\u5a92\u3092\u7528\u3044\u305f3-\u30cb\u30c8\u30ed\u30af\u30de\u30ea\u30f3\u306e\u4e0d\u6589Diels\u2013Alder\u53cd\u5fdc\u3068\u901f\u5ea6\u8ad6\u7684\u5149\u5b66\u5206\u5272\u300d<br>\u5742\u5009\u5f70\uff0c\u85e4\u4e95\u88d5\u5927\uff0c\u4e2d\u5c3e\u4eae\u592a\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u6e9d\u53e3\u7384\u6a39<br>\u7b2c11\u56de\u6709\u6a5f\u89e6\u5a92\u30b7\u30f3\u30dd\u30b8\u30a6\u30e0\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6771\u4eac\uff0c\u5b66\u7fd2\u9662\u5927\u5b66\uff0c2018\u5e7412\u67083\u65e5\uff0c4\u65e5<\/li>\n<\/ol>\n\n\n\n<ol class=\"wp-block-list\">\n<li>\u300c\u30b2\u30e9\u30cb\u30eb\u8a98\u5c0e\u4f53\u306e\u30d0\u30a4\u30aa\u30df\u30e1\u30c6\u30a3\u30c3\u30af\u306a\u30d6\u30ed\u30e2\u74b0\u5316\u53cd\u5fdc\u306b\u6709\u52b9\u306a\u30c1\u30aa\u30a6\u30ec\u30a2\u89e6\u5a92\u300d<br>\u5742\u5009\u5f70\uff0c\u5bfa\u5d0e\u7f8e\u5e78\uff0c\u5869\u672c\u5553\u4e00\uff0c\u6e9d\u53e3\u7384\u6a39<br>\u7b2c60\u56de\u5929\u7136\u6709\u6a5f\u5316\u5408\u7269\u8a0e\u8ad6\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u4e45\u7559\u7c73\u30b7\u30c6\u30a3\u30fc\u30d7\u30e9\u30b6\uff0c2018\u5e749\u670826\u301c28\u65e5\uff0cP2-19<\/li>\n<\/ol>\n\n\n\n<p><\/p>\n\n\n\n<p style=\"font-size:20px\"><strong>2017\u5e74\u5ea6<\/strong><\/p>\n\n\n\n<ol start=\"11\" class=\"wp-block-list\">\n<li>\u300c\u30e6\u30ba\u30ea\u30df\u30f3\u985e\u306e\u70ad\u7d20\u9aa8\u683c\u306e\u5408\u6210\u7814\u7a76 (Synthetic Studies of Core Carbon Framework of Yuzurimine-type Alkaloids)\u300d<br>\u4e2d\u91cd\u96c4\u4e00\uff0c\u5409\u4fe1\u62d3\u54c9\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c98\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u7406\u5de5\u5b66\u90e8\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2018\u5e743\u670822\u65e5\uff0c3D2-06<\/li>\n<\/ol>\n\n\n\n<ol start=\"10\" class=\"wp-block-list\">\n<li>\u300c\u30a2\u30eb\u30c6\u30df\u30b7\u30b8\u30f3\u985e\u306e\u5408\u6210\u7814\u7a76 (Synthetic Studies of Altemicidin-type Alkaloids)\u300d<br>\u6c38\u6613\u674f\u83dc\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c98\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u7406\u5de5\u5b66\u90e8\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2018\u5e743\u670822\u65e5\uff0c3D2-05<\/li>\n<\/ol>\n\n\n\n<ol start=\"9\" class=\"wp-block-list\">\n<li>\u300cN-\u30a2\u30bb\u30c1\u30eb\u30b3\u30eb\u30d2\u30ce\u30fc\u30eb\u306e\u5408\u6210\u7814\u7a76 (Synthetic Studies of N-Acetylcolchinol)\u300d<br>\u4e2d\u91ce\u967d\u4e00\u90ce\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c98\u6625\u5b63\u5e74\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u7406\u5de5\u5b66\u90e8\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2018\u5e743\u670821\u65e5\uff0c2PB-012<\/li>\n<\/ol>\n\n\n\n<ol start=\"8\" class=\"wp-block-list\">\n<li>\u300c\u30b2\u30e9\u30cb\u30eb\u8a98\u5c0e\u4f53\u306e\u30d6\u30ed\u30e2\u74b0\u5316\u53cd\u5fdc\u306b\u6709\u52b9\u306a\u30c1\u30aa\u30a6\u30ec\u30a2\u304a\u3088\u3073\u30c1\u30aa\u30ea\u30f3\u9178\u30a2\u30df\u30c9\u89e6\u5a92 (Thiourea and Thiophosphoric Amides as Highly Active Catalysts for Selective Bromocyclization of Geranyl Derivatives)\u300d<br>\u5bfa\ufa11\u7f8e\u5e78\uff0c\u5869\u672c\u5553\u4e00\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c98\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u7406\u5de5\u5b66\u90e8\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2018\u5e743\u670820\u65e5\uff0c1H5-13<\/li>\n<\/ol>\n\n\n\n<ol start=\"7\" class=\"wp-block-list\">\n<li>\u300c\u30ad\u30e9\u30eb\u306a\u30d6\u30ec\u30f3\u30b9\u30c6\u30c3\u30c9\u9178\u89e6\u5a92\u3092\u7528\u3044\u305f\u03b1-\u7f6e\u63db\u03b1-\u30cb\u30c8\u30ed\u30e9\u30af\u30c8\u30f3\u306e\u901f\u5ea6\u8ad6\u7684\u5149\u5b66\u5206\u5272 (Kinetic Resolution of \u03b1-Substituted \u03b1-Nitrolactones Promoted by Br\u00f8nsted Acid Catalysts) \u300d<br>\u4e2d\u5c3e\u4eae\u592a\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c98\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u7406\u5de5\u5b66\u90e8\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2018\u5e743\u670820\u65e5\uff0c1H5-12<\/li>\n<\/ol>\n\n\n\n<ol start=\"6\" class=\"wp-block-list\">\n<li>\u300c\u30ac\u30bf\u30b9\u30bf\u30c1\u30f3\u3092\u30ea\u30fc\u30c9\u5316\u5408\u7269\u3068\u3057\u305f\u03b3-\u30c1\u30e5\u30fc\u30d6\u30ea\u30f3\u7279\u7570\u7684\u963b\u5bb3\u5264\u306e\u958b\u767a\u7814\u7a76 \u300d<br>\u65e9\u5ddd\u4e00\u90ce\uff0c\u7551\u4e2d\u5927\u6210\uff0c \u5869\u7530\u79c0\u4e5f\uff0c\u77e5\u5ff5\u62d3\u5b9f\uff0c\u6075\u6bd4\u5bff\u6625\u83dc\uff0c\u81fc\u4e95\u5065\u90ce\uff0c\u6728\u8d8a\u82f1\u592b\uff0c\u5742\u5009\u5f70<br>\u7b2c35\u56de\u30e1\u30c7\u30a3\u30b7\u30ca\u30eb\u30b1\u30df\u30b9\u30c8\u30ea\u30fc\u30b7\u30f3\u30dd\u30b8\u30a6\u30e0\u3000\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u540d\u53e4\u5c4b\u5927\u5b66\u8c4a\u7530\u8b1b\u5802\uff0c2017\u5e7410\u670825\u65e5\u301c27\u65e5\uff0c1P-083<\/li>\n<\/ol>\n\n\n\n<ol start=\"5\" class=\"wp-block-list\">\n<li>\u300c\u30e6\u30ba\u30ea\u30cf\u30a2\u30eb\u30ab\u30ed\u30a4\u30c9\u30fb\u30e6\u30ba\u30ea\u30df\u30f3\u985e\u306e\u5408\u6210\u7814\u7a76\u300d<br>\u65e9\u5ddd\u4e00\u90ce\uff0c\u6c60\u7530\u5c06\u898f\uff0c\u65b0\u4e95\u7530\u6075\u4ecb\uff0c\u4e2d\u91cd\u96c4\u4e00\uff0c\u6c38\u6613\u674f\u83dc\uff0c\u91ce\u6751\u7d17\u5e0c\uff0c\u9f4a\u85e4\u5553\u592a\uff0c\u6728\u8d8a\u82f1\u592b\uff0c\u5742\u5009\u5f70<br>\u7b2c59\u56de\u5929\u7136\u6709\u6a5f\u5316\u5408\u7269\u8a0e\u8ad6\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u308f\u304f\u308f\u304f\u30db\u30ea\u30c7\u30fc\u30db\u30fc\u30eb\uff08\u672d\u5e4c\u5e02\u6c11\u30db\u30fc\u30eb\uff09\uff0c2017\u5e749\u670820\u65e5\u301c22\u65e5\uff0cP-33<\/li>\n<\/ol>\n\n\n\n<ol start=\"4\" class=\"wp-block-list\">\n<li>\u300c\u30eb\u30a4\u30b9\u9178\u304a\u3088\u3073\u30d6\u30ec\u30f3\u30b9\u30c6\u30c3\u30c9\u9178\u89e6\u5a92\u3092\u7528\u3044\u308b\u4e0d\u98fd\u548c2\u7d1a\u30a2\u30eb\u30b3\u30fc\u30eb\u306e\u5206\u5b50\u5185\u30cf\u30ed\u30a8\u30fc\u30c6\u30eb\u74b0\u5316\u53cd\u5fdc\u306e\u691c\u8a0e\u300d<br>\u5869\u672c\u5553\u4e00\uff0c\u5742\u5009\u5f70<br>\u7b2c33\u56de\u82e5\u624b\u5316\u5b66\u8005\u306e\u305f\u3081\u306e\u5316\u5b66\u9053\u5834\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u9ce5\u53d6\u770c\u9ce5\u53d6\u5e02 \u30ec\u30fc\u30af\u5927\u6a39\uff0c2017\u5e749\u67081\u65e5\uff0c2\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"3\" class=\"wp-block-list\">\n<li>\u300c\u30ad\u30e9\u30eb\u6709\u6a5f\u30a2\u30f3\u30e2\u30cb\u30a6\u30e0\u5869\u89e6\u5a92\u3092\u7528\u3044\u305f\u30cb\u30c8\u30ed\u30f3\u3068\u03b1-\u30a2\u30b7\u30ed\u30ad\u30b7\u30a2\u30af\u30ed\u30ec\u30a4\u30f3\u3068\u306e\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u76841,3-\u53cc\u6975\u5b50\u74b0\u5316\u4ed8\u52a0\u53cd\u5fdc\u306e\u958b\u767a\u300d<br>\u9b3c\u7ae5\u3061\u3072\u308d\uff0c\u5742\u5009\u5f70<br>\u7b2c33\u56de\u82e5\u624b\u5316\u5b66\u8005\u306e\u305f\u3081\u306e\u5316\u5b66\u9053\u5834\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u9ce5\u53d6\u770c\u9ce5\u53d6\u5e02 \u30ec\u30fc\u30af\u5927\u6a39\uff0c2017\u5e749\u67081\u65e5\uff0c2\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"2\" class=\"wp-block-list\">\n<li>\u201cTotal Synthesis of Manzacidins A and C Based on Diastereoselective Hydroxymethylation of Chiral Nitroalkanes\"<br>Yuya Araki, Mizuho Tanioka, Natsumi Miyoshi, Takayuki Kudoh, Akira Sakakura<br>International Symposium on Pure &amp; Applied Chemistry (ISPAC) 2017, oral presentation, ORG67<br>Hotel Continental Saigon, Ho Chi Minh City, Vietnam, June 8-10, 2017<\/li>\n<\/ol>\n\n\n\n<ol class=\"wp-block-list\">\n<li>\"Biomimetic Cyclization of 3,5-Diketoesters: Application to Total Synthesis of Cyercene A, an \u03b1-Methoxy-\u03b3-Pyrone-Containing Polypropionate\"<br>Akira Sakakura<br>International Symposium on Pure &amp; Applied Chemistry (ISPAC) 2017, invited lecture, oral presentation, ORG42<br>Hotel Continental Saigon, Ho Chi Minh City, Vietnam, June 8-10, 2017<\/li>\n<\/ol>\n\n\n\n<p><\/p>\n\n\n\n<p style=\"font-size:20px\"><strong>2016\u5e74\u5ea6<\/strong><\/p>\n\n\n\n<ol start=\"10\" class=\"wp-block-list\">\n<li>\u300c3,5-\u30b8\u30b1\u30c8\u30a8\u30b9\u30c6\u30eb\u306e\u5206\u5b50\u5185\u30a8\u30b9\u30c6\u30eb\u4ea4\u63db\u53cd\u5fdc\u3092\u7528\u3044\u305f\u30b5\u30a4\u30a8\u30eb\u30bb\u30f3A\u306e\u5168\u5408\u6210 (Total synthesis of cyercene A using intramolecular transesterification reaction of 3,5-diketoester as a key step)\u300d<br>\u6069\u7530\u958b\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c97\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6176\u61c9\u7fa9\u587e\u5927\u5b66\u3000\u65e5\u5409\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2017\u5e743\u670818\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"9\" class=\"wp-block-list\">\n<li>\u300c\u30ad\u30e9\u30eb\u6709\u6a5f\u30a2\u30f3\u30e2\u30cb\u30a6\u30e0\u5869\u89e6\u5a92\u3092\u7528\u3044\u305f\u30cb\u30c8\u30ed\u30f3\u3068\u03b1-\u30a2\u30b7\u30ed\u30ad\u30b7\u30a2\u30af\u30ed\u30ec\u30a4\u30f3\u3068\u306e\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u76841,3-\u53cc\u6975\u5b50\u74b0\u5316\u4ed8\u52a0\u53cd\u5fdc (Enantioselective 1,3-Dipolar Cycloaddition of \u03b1-Acyloxyacroleins with Nitrones Catalyzed by Chiral Organoammonium salts)\u300d<br>\u9b3c\u7ae5\u3061\u3072\u308d\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c97\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6176\u61c9\u7fa9\u587e\u5927\u5b66\u3000\u65e5\u5409\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2017\u5e743\u670816\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"8\" class=\"wp-block-list\">\n<li>\u300c\u30ad\u30e9\u30eb\u306a\u4e9c\u30ea\u30f3\u9178\u30a8\u30b9\u30c6\u30eb\u3068\u30ad\u30e9\u30eb\u306a\u30a6\u30ec\u30a2\u3092\u7d44\u307f\u5408\u308f\u305b\u305f\u6709\u6a5f\u5206\u5b50\u89e6\u5a92\u306b\u3088\u308b2-\u30b2\u30e9\u30cb\u30eb\u30d5\u30a7\u30ce\u30fc\u30eb\u306e\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u7684\u30d6\u30ed\u30e2\u74b0\u5316\u53cd\u5fdc (Enantioselective Bromocyclization of 2-Geranylphenols Promoted by Chiral Phosphite-Chiral Urea Combined Catalysts)\u300d<br>\u5bfa\u5d0e\u7f8e\u5e78\uff0c\u5f35\u5922\u83ef\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c97\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6176\u61c9\u7fa9\u587e\u5927\u5b66\u3000\u65e5\u5409\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2017\u5e743\u670816\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"7\" class=\"wp-block-list\">\n<li>\u300cn-\u30ab\u30c1\u30aa\u30f3\u89e6\u5a92\u3092\u7528\u3044\u308b\u30a2\u30ea\u30eb\u30b7\u30e9\u30f3\u306e\u03b1-\u30b1\u30c8\u30a8\u30b9\u30c6\u30eb\u306b\u5bfe\u3059\u308b\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u7684\u6c42\u6838\u4ed8\u52a0\u53cd\u5fdc (Enantioselective Addition of Allylic Silanes with \u03b1\u2212Ketoesters Induced by n-Cation Catalyst)\u300d<br>\u4e39\u7fbd\u7950\u592a\u6717\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c97\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6176\u61c9\u7fa9\u587e\u5927\u5b66\u3000\u65e5\u5409\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2017\u5e743\u670816\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"6\" class=\"wp-block-list\">\n<li>\u300c\u30b8\u30a2\u30b9\u30c6\u30ec\u30aa\u9078\u629e\u7684\u30d2\u30c9\u30ed\u30ad\u30b7\u30e1\u30c1\u30eb\u5316\u3092\u9375\u53cd\u5fdc\u3068\u3059\u308b\u30de\u30f3\u30b6\u30b7\u30b8\u30f3A\u304a\u3088\u3073C\u306e\u5168\u5408\u6210 (Total Synthesis of Manzacidins A and C Based on Diastereoselective Hydroxymethylation of Chiral Nitroalkanes)\u300d<br>\u8352\u6728\u96c4\u4e5f\uff0c\u8c37\u5ca1\u745e\u6b69\uff0c\u4e09\u597d\u590f\u7f8e\uff0c\u5de5\u85e4\u5b5d\u5e78\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c97\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6176\u61c9\u7fa9\u587e\u5927\u5b66\u3000\u65e5\u5409\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2017\u5e743\u670816\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"5\" class=\"wp-block-list\">\n<li>\u300c\u5929\u7136\u7269\u5168\u5408\u6210\u3092\u8d77\u70b9\u3068\u3057\u305f\u751f\u4f53\u6a5f\u80fd\u5206\u5b50\u306e\u958b\u767a\u7814\u7a76\u300d<br>\u65e9\u5ddd\u4e00\u90ce<br>\u7b2c27\u56de\u795e\u5948\u5ddd\u5927\u5b66\u5e73\u585a\u30b7\u30f3\u30dd\u30b8\u30a6\u30e0\u300c\u3082\u306e\u3065\u304f\u308a\u306e\u6700\u524d\u7dda\u2014\u30de\u30c6\u30ea\u30a2\u30eb\u304b\u3089\u30d0\u30a4\u30aa\u30b5\u30a4\u30a8\u30f3\u30b9\u307e\u3067\u300d\uff0c\u62db\u5f85\u8b1b\u6f14\uff0c\u795e\u5948\u5ddd\u5927\u5b66\u6e58\u5357\u3072\u3089\u3064\u304b\u30ad\u30e3\u30f3\u30d1\u30b911\u53f7\u9928\u30b5\u30fc\u30ab\u30e0\u30db\u30fc\u30eb\uff0c2017\u5e743\u67084\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"4\" class=\"wp-block-list\">\n<li>\u300c\u30b8\u30a2\u30b9\u30c6\u30ec\u30aa\u9078\u629e\u7684\u30d2\u30c9\u30ed\u30ad\u30b7\u30e1\u30c1\u30eb\u5316\u53cd\u5fdc\u3092\u9375\u5de5\u7a0b\u3068\u3059\u308b\u30de\u30f3\u30b6\u30b7\u30b8\u30f3 A, C \u306e\u5408\u6210\u7814\u7a76\u300d<br>\u8352\u6728\u96c4\u4e5f\uff0c\u4e09\u597d\u590f\u7f8e\uff0c\u8c37\u5ca1\u745e\u6b69\uff0c\u5de5\u85e4\u5b5d\u5e78\uff0c\u5742\u5009\u5f70<br>2016\u5e74\u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u9999\u5ddd\u5927\u5b66\u5e78\u753a\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2016\u5e7411\u67086\u65e5<\/li>\n<\/ol>\n\n\n\n<p>3.\u300c\u30ad\u30e9\u30eb\u306a\u30cb\u30c8\u30ed\u30a2\u30eb\u30ab\u30f3\u306b\u5bfe\u3059\u308b\u30b8\u30a2\u30b9\u30c6\u30ec\u30aa\u9078\u629e\u7684\u30d2\u30c9\u30ed\u30ad\u30b7\u30e1\u30c1\u30eb\u5316\u53cd\u5fdc\u3092\u9375\u5de5\u7a0b\u3068\u3059\u308b\u30de\u30f3\u30b6\u30b7\u30b8\u30f3\u985e\u306e\u5408\u6210\u7814\u7a76\u300d<br>\u5de5\u85e4\u5b5d\u5e78\uff0c\u4e09\u597d\u590f\u7f8e\uff0c\u8352\u6728\u96c4\u4e5f\uff0c\u5742\u5009\u5f70<br>\u7b2c58\u56de\u5929\u7136\u6709\u6a5f\u5316\u5408\u7269\u8a0e\u8ad6\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u6771\u5317\u5927\u5b66\u767e\u5468\u5e74\u8a18\u5ff5\u4f1a\u9928\u5ddd\u5185\u8429\u30db\u30fc\u30eb\u30fb\u5ddd\u5185\u5317\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2016\u5e749\u670814\u65e5\uff0cP-25<\/p>\n\n\n\n<ol start=\"2\" class=\"wp-block-list\">\n<li>\u300c\u4e09\u7f6e\u63db\u30cb\u30c8\u30ed\u30a2\u30eb\u30b1\u30f3\u306b\u5bfe\u3059\u308b\u7acb\u4f53\u9078\u629e\u7684\u74b0\u5316\u4ed8\u52a0\u53cd\u5fdc\u306b\u3088\u308b\u30a2\u30df\u30ce\u57fa\u7d50\u5408\u4e0d\u6589\u56db\u7d1a\u70ad\u7d20\u306e\u69cb\u7bc9\u300d<br>\u4e2d\u5c3e\u4eae\u592a\uff0c\u5de5\u85e4\u5b5d\u5e78\uff0c\u5742\u5009\u5f70<br>\u7b2c32\u56de\u82e5\u624b\u5316\u5b66\u8005\u306e\u305f\u3081\u306e\u5316\u5b66\u9053\u5834\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u611b\u5a9b\u770c\u677e\u5c71\u5e02\u306b\u304e\u305f\u3064\u4f1a\u9928\uff0c2016\u5e748\u670825, 26\u65e5<\/li>\n<\/ol>\n\n\n\n<ol class=\"wp-block-list\">\n<li>\u300c\u03b1-\u30b1\u30c8\u30a8\u30b9\u30c6\u30eb\u306b\u5bfe\u3059\u308b\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u7684\u306a\u6c42\u6838\u4ed8\u52a0\u53cd\u5fdc\u3092\u5229\u7528\u3057\u305f\u4e0d\u6589\u56db\u7d1a\u70ad\u7d20\u69cb\u7bc9\u6cd5\u306e\u958b\u767a\u300d<br>\u4e39\u7fbd\u7950\u592a\u6717\uff0c\u5742\u5009\u5f70<br>\u7b2c32\u56de\u82e5\u624b\u5316\u5b66\u8005\u306e\u305f\u3081\u306e\u5316\u5b66\u9053\u5834\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u611b\u5a9b\u770c\u677e\u5c71\u5e02\u306b\u304e\u305f\u3064\u4f1a\u9928\uff0c2016\u5e748\u670825, 26\u65e5<\/li>\n<\/ol>\n\n\n\n<p><\/p>\n\n\n\n<p style=\"font-size:20px\"><strong>2015\u5e74\u5ea6<\/strong><\/p>\n\n\n\n<ol start=\"22\" class=\"wp-block-list\">\n<li>\u300c3,5-\u30b8\u30b1\u30c8\u30a8\u30b9\u30c6\u30eb\u306e\u5206\u5b50\u5185\u30a8\u30b9\u30c6\u30eb\u4ea4\u63db\u53cd\u5fdc\u306b\u3088\u308b\u03b1-\u30e1\u30c8\u30ad\u30b7-\u03b3-\u30d4\u30ed\u30f3\u5316\u5408\u7269\u306e\u5408\u6210\u7814\u7a76 (Development of Intramolecular Transesterification Reaction of 3,5-Diketoester for Synthesis of \u03b1-methoxy-\u03b3-pyrone compounds)\u300d<br>\u6069\u7530\u958b\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c96\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0cATP\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u540c\u5fd7\u793e\u5927\u5b66\u3000\u4eac\u7530\u8fba\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2016\u5e743\u670824\u65e5\uff0c26\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"21\" class=\"wp-block-list\">\n<li>\u300c\u30b0\u30e9\u30b8\u30aa\u30d3\u30a2\u30cb\u30f3A\u3092\u30ea\u30fc\u30c9\u5316\u5408\u7269\u3068\u3057\u305f\u03b3-\u30c1\u30e5\u30fc\u30d6\u30ea\u30f3\u7279\u7570\u7684\u963b\u5bb3\u5264\u306e\u958b\u767a\u7814\u7a76 (Structure\u2013Activity Relationship Study of Glaziovianin A for the Development of \u03b3-Tubulin-Specific Inhibitor)\u300d<br>\u7551\u4e2d\u5927\u6210\uff0c\u5869\u7530\u79c0\u4e5f\uff0c\u77e5\u5ff5\u62d3\u5b9f\uff0c\u6075\u6bd4\u5bff\u6625\u83dc\uff0c\u81fc\u4e95\u5065\u90ce\uff0c\u6728\u8d8a\u82f1\u592b\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c96\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u540c\u5fd7\u793e\u5927\u5b66\u3000\u4eac\u7530\u8fba\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2016\u5e743\u670826\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"20\" class=\"wp-block-list\">\n<li>\u300c\u30a4\u30f3\u30c9\u30fc\u30eb\u7d50\u54081,6-\u30b8\u30a4\u30f3\u306e\u5206\u5b50\u5185\u30c7\u30d2\u30c9\u30edDiels-Alder\u53cd\u5fdc\u306b\u3088\u308b\u65b0\u898f\u7f6e\u63db\u30ab\u30eb\u30d0\u30be\u30fc\u30eb\u5408\u6210\u6cd5\u306e\u958b\u767a (Development of Intramolecular Dehydro Diels-Alder Reaction of Indolyl-1,6-diynes for the Synthesis of Substituted Carbazoles)\u300d<br>\u85e4\u6fa4\u7fd4\uff0c\u5de5\u85e4\u5b5d\u5e78\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c96\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0cATP\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u540c\u5fd7\u793e\u5927\u5b66\u3000\u4eac\u7530\u8fba\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2016\u5e743\u670824\u65e5\uff0c25\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"19\" class=\"wp-block-list\">\n<li>\u300c\u4e09\u7f6e\u63db\u30cb\u30c8\u30ed\u30a2\u30eb\u30b1\u30f3\u306e\u4e0d\u6589Diels-Alder\u53cd\u5fdc\u306b\u6709\u52b9\u306a\u30ad\u30e9\u30eb\u30d6\u30ec\u30f3\u30b9\u30c6\u30c3\u30c9\u9178\u89e6\u5a92\u306e\u7cbe\u5bc6\u8a2d\u8a08 (Design of Chiral Br\u00f8nsted Acid Catalysts for Asymmetric Diels-Alder Reaction of Trisubstituted Nitroalkenes)\u300d<br>\u85e4\u4e95\u88d5\u5927\uff0c\u5de5\u85e4\u5b5d\u5e78\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c96\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0cATP\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u540c\u5fd7\u793e\u5927\u5b66\u3000\u4eac\u7530\u8fba\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2016\u5e743\u670824\u65e5\uff0c25\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"18\" class=\"wp-block-list\">\n<li>\u300c\u30e6\u30ba\u30ea\u30cf\u30a2\u30eb\u30ab\u30ed\u30a4\u30c9\u30fb\u30e6\u30ba\u30ea\u30df\u30f3\u985e\u306e\u8907\u7d20\u74b0\u90e8\u5206\u306e\u5408\u6210\u7814\u7a76 (Synthetic Study of a Heterocyclic Portion of Yuzurimine-type Alkaloids)\u300d<br>\u6c60\u7530\u5c06\u898f\uff0c\u91ce\u6751\u7d17\u5e0c\uff0c\u658e\u85e4\u5553\u592a\uff0c\u6728\u8d8a\u82f1\u592b\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c96\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u540c\u5fd7\u793e\u5927\u5b66\u3000\u4eac\u7530\u8fba\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2016\u5e743\u670824\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"17\" class=\"wp-block-list\">\n<li>\u300c\u30b8\u30a2\u30b9\u30c6\u30ec\u30aa\u9078\u629e\u7684\u30d2\u30c9\u30ed\u30ad\u30b7\u30e1\u30c1\u30eb\u5316\u3092\u9375\u53cd\u5fdc\u3068\u3059\u308b\u30de\u30f3\u30b6\u30b7\u30b8\u30f3B\u306e\u5408\u6210\u7814\u7a76 (Synthetic Study of Manzacidin B Based on Diastereoselective Hydroxymethylation)\u300d<br>\u4e09\u597d\u590f\u7f8e\uff0c\u8352\u6728\u96c4\u4e5f\uff0c\u5de5\u85e4\u5b5d\u5e78\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c96\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u540c\u5fd7\u793e\u5927\u5b66\u3000\u4eac\u7530\u8fba\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2016\u5e743\u670824\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"16\" class=\"wp-block-list\">\n<li>\u201cSynthetic studies of manzacidins A-C based on diastereoselective hydroxymethylation of chiral nitro compounds\u201d<br>Akira Sakakura,* Natsumi Miyoshi, Takayuki Kudoh<br>The 2015 International Chemical Congress of Pacific Basin Societies (PAC CHEM\u2122, Pacifichem 2015), Honolulu, Hawaii, USA, December 19, 2015, ORGN 2384, Natural Product-based Drug Discovery (#66)<\/li>\n<\/ol>\n\n\n\n<ol start=\"15\" class=\"wp-block-list\">\n<li>\u300c\u6297\u816b\u760d\u6d3b\u6027\u7269\u8cea\u30b0\u30e9\u30b8\u30aa\u30d3\u30a2\u30cb\u30f3A\u306e\u69cb\u9020\u6d3b\u6027\u76f8\u95a2\u7814\u7a76\u300d<br>\u7551\u4e2d\u5927\u6210\uff0c\u5869\u7530\u79c0\u4e5f\uff0c\u77e5\u5ff5\u62d3\u5b9f\uff0c\u81fc\u4e95\u5065\u90ce\uff0c\u6728\u8d8a\u82f1\u592b\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>2015\u5e74\u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2015\u5e7411\u670815\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"14\" class=\"wp-block-list\">\n<li>\u300c\u9396\u72b6\u524d\u99c6\u4f53\u306e\u5206\u5b50\u5185\u30a8\u30b9\u30c6\u30eb\u4ea4\u63db\u53cd\u5fdc\u3092\u5229\u7528\u3057\u305f\u03b3-\u30d4\u30ed\u30f3\u5316\u5408\u7269\u306e\u5408\u6210\u7814\u7a76\u300d<br>\u6069\u7530\u958b\uff0c\u5742\u5009\u5f70<br>2015\u5e74\u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2015\u5e7411\u670815\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"13\" class=\"wp-block-list\">\n<li>\u300c\u8fbb\u2013Trost\u53cd\u5fdc\u306b\u3088\u308b\u30e1\u30bd\u30b8\u30aa\u30fc\u30eb\u8a98\u5c0e\u4f53\u306e\u4e0d\u6589\u975e\u5bfe\u79f0\u5316\u53cd\u5fdc\u3092\u9375\u53cd\u5fdc\u3068\u3057\u305f(\u2013)-\u30d9\u30eb\u30ab\u30ed\u30fc\u30eb\u306e\u5408\u6210\u7814\u7a76\u300d<br>\u4e09\u57a3\u8056\u4e5f\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>2015\u5e74\u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2015\u5e7411\u670815\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"12\" class=\"wp-block-list\">\n<li>\u300c\u30e6\u30ba\u30ea\u30df\u30f3\u985e\u306e\u8907\u7d20\u74b0\u90e8\u5206\u306e\u5408\u6210\u7814\u7a76\u300d<br>\u6c60\u7530\u5c06\u898f\uff0c\u91ce\u6751\u7d17\u5e0c\uff0c\u658e\u85e4\u5553\u592a\uff0c\u6728\u8d8a\u82f1\u592b\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>2015\u5e74\u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2015\u5e7411\u670815\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"11\" class=\"wp-block-list\">\n<li>\u300c\u30b8\u30a2\u30b9\u30c6\u30ec\u30aa\u9078\u629e\u7684Henry\u53cd\u5fdc\u3092\u9375\u53cd\u5fdc\u3068\u3059\u308b\u30de\u30f3\u30b6\u30b7\u30b8\u30f3\uff22\u306e\u5168\u5408\u6210\u7814\u7a76\u300d<br>\u4e09\u597d\u590f\u7f8e\uff0c\u8352\u6728\u96c4\u4e5f\uff0c\u5de5\u85e4\u5b5d\u5e78\uff0c\u5742\u5009\u5f70<br>2015\u5e74\u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2015\u5e7411\u670815\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"10\" class=\"wp-block-list\">\n<li>\u300c\u4e09\u7f6e\u63db\u30cb\u30c8\u30ed\u30a2\u30eb\u30b1\u30f3\u3092\u7528\u3044\u305f\u7acb\u4f53\u9078\u629e\u7684Diels-Alder\u53cd\u5fdc\u306e\u958b\u767a\u300d<br>\u85e4\u4e95\u88d5\u5927\uff0c\u5de5\u85e4\u5b5d\u5e78\uff0c\u5742\u5009\u5f70<br>2015\u5e74\u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2015\u5e7411\u670815\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"9\" class=\"wp-block-list\">\n<li>\u300c\u30a4\u30f3\u30c9\u30fc\u30eb\u7d50\u54081,6-\u30b8\u30a4\u30f3\u306e\u5206\u5b50\u5185\u30c7\u30d2\u30c9\u30edDiels-Alder\u53cd\u5fdc\u306b\u3088\u308b\u30ab\u30eb\u30d0\u30be\u30fc\u30eb\u5408\u6210\u300d<br>\u85e4\u6fa4\u7fd4\uff0c\u5de5\u85e4\u5b5d\u5e78\uff0c\u5742\u5009\u5f70<br>2015\u5e74\u65e5\u672c\u5316\u5b66\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8\u5927\u4f1a\uff0c\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2015\u5e7411\u670815\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"8\" class=\"wp-block-list\">\n<li>\u300c\u65b0\u898f\u5206\u5b50\u5185\u74b0\u5316\u4ed8\u52a0\u53cd\u5fdc\u306e\u958b\u767a\u3068\u6709\u6a5f\u5408\u6210\u5316\u5b66\u3092\u57fa\u76e4\u3068\u3059\u308b\u751f\u7269\u6d3b\u6027\u7269\u8cea\u306e\u5275\u51fa\u300d<br>\u5de5\u85e4\u5b5d\u5e78<br>\u5e73\u621027\u5e74\u5ea6\u652f\u90e8\u5968\u52b1\u8cde\u53d7\u8cde\u8005\u8b1b\u6f14\uff0c\u5ca1\u5c71\u5927\u5b66\u5de5\u5b66\u90e81\u53f7\u9928\u5927\u8b1b\u7fa9\u5ba4\uff0c2015\u5e7411\u670814\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"7\" class=\"wp-block-list\">\n<li>\"A Short Entry to 3,5-Disubstituted Piperazinones Based on Aza-Michael Addition of \u03b1-Amino Esters to Nitroalkenes\"<br>Akira Sakakura,* Takayuki Kudoh, Seiji Isoyama, and Sachiko Kagimoto<br>The 10th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-10), invited lecture, 85 SKY TOWER HOTEL, KaoHsiung, Taiwan, November 2 (Mon) to November 5 (Thu), 2015<\/li>\n<\/ol>\n\n\n\n<ol start=\"6\" class=\"wp-block-list\">\n<li>\u300c\u30e6\u30ba\u30ea\u30cf\u30a2\u30eb\u30ab\u30ed\u30a4\u30c9\u30fb\u30e6\u30ba\u30ea\u30df\u30f3\u985e\u306e\u8907\u7d20\u74b0\u90e8\u5206\u306e\u5408\u6210\u7814\u7a76\u300d<br>\u6c60\u7530\u5c06\u898f\uff0c\u91ce\u6751\u7d17\u5e0c\uff0c\u658e\u85e4\u5553\u592a\uff0c\u6728\u8d8a\u82f1\u592b\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>\u7b2c31\u56de\u82e5\u624b\u5316\u5b66\u8005\u306e\u305f\u3081\u306e\u5316\u5b66\u9053\u5834\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u6de1\u8def\u5922\u821e\u53f0\u56fd\u969b\u4f1a\u8b70\u5834\uff0c2015\u5e748\u670827, 28\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"5\" class=\"wp-block-list\">\n<li>\u300c\u30a4\u30f3\u30c9\u30fc\u30eb\u7d50\u54081,6-\u30b8\u30a4\u30f3\u3092\u7528\u3044\u305fDehydro Diels\u2013Alder\u53cd\u5fdc\u306e\u691c\u8a0e\u300d<br>\u85e4\u6fa4\u7fd4\uff0c\u5de5\u85e4\u5b5d\u5e78\uff0c\u5742\u5009\u5f70<br>\u7b2c31\u56de\u82e5\u624b\u5316\u5b66\u8005\u306e\u305f\u3081\u306e\u5316\u5b66\u9053\u5834\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u6de1\u8def\u5922\u821e\u53f0\u56fd\u969b\u4f1a\u8b70\u5834\uff0c2015\u5e748\u670827, 28\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"4\" class=\"wp-block-list\">\n<li>\u300c\u8fbb\u2013Trost\u53cd\u5fdc\u306b\u3088\u308b\u4e0d\u6589\u975e\u5bfe\u79f0\u5316\u53cd\u5fdc\u3092\u9375\u53cd\u5fdc\u3068\u3057\u305f(\u2013)-\u30d9\u30eb\u30ab\u30ed\u30fc\u30eb\u306e\u5408\u6210\u7814\u7a76\u300d<br>\u4e09\u57a3\u8056\u4e5f\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>\u7b2c31\u56de\u82e5\u624b\u5316\u5b66\u8005\u306e\u305f\u3081\u306e\u5316\u5b66\u9053\u5834\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u6de1\u8def\u5922\u821e\u53f0\u56fd\u969b\u4f1a\u8b70\u5834\uff0c2015\u5e748\u670827, 28\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"3\" class=\"wp-block-list\">\n<li>\u300c\u9ad8\u5ea6\u306b\u7e2e\u74b0\u3057\u305f\u5929\u7136\u7269\u306e\u5408\u6210\u7814\u7a76\u300d<br>\u65e9\u5ddd\u4e00\u90ce<br>\u7b2c31\u56de\u82e5\u624b\u5316\u5b66\u8005\u306e\u305f\u3081\u306e\u5316\u5b66\u9053\u5834\uff0c\u5e2b\u7bc4\u8b1b\u6f14\uff0c\u6de1\u8def\u5922\u821e\u53f0\u56fd\u969b\u4f1a\u8b70\u5834\uff0c2015\u5e748\u670827, 28\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"2\" class=\"wp-block-list\">\n<li>\u300c\u9ad8\u5ea6\u306b\u7e2e\u74b0\u3057\u305f\u5929\u7136\u7269\u306e\u5408\u6210\u7814\u7a76\u300d<br>\u65e9\u5ddd\u4e00\u90ce<br>\u5ca1\u5c71\u5927\u5b66\u7570\u5206\u91ce\u878d\u5408\u7814\u7a76\u80b2\u6210\u652f\u63f4\u4e8b\u696d\u300c\u6709\u6a5f\u5408\u6210\u3092\u57fa\u76e4\u3068\u3057\u305f\u751f\u4f53\u6a5f\u80fd\u5236\u5fa1\u5206\u5b50\u306e\u5275\u88fd\u300d\u7b2c2\u56de\u8b1b\u6f14\u4f1a\uff0c\u5ca1\u5c71\u5927\u5b66\u7406\u5b66\u90e8\uff0c2015\u5e747\u670831\u65e5<\/li>\n<\/ol>\n\n\n\n<ol class=\"wp-block-list\">\n<li>\u300c\u30cf\u30ed\u30b2\u30f3\u7d50\u5408\u306b\u3088\u308b\u30e8\u30a6\u7d20\u5316\u5264\u306e\u6d3b\u6027\u5316\u3092\u9375\u3068\u3059\u308b\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u7684\u30e8\u30fc\u30c9\u30e9\u30af\u30c8\u30f3\u5316\u53cd\u5fdc\u306e\u958b\u767a\u300d<br>\u5742\u5009\u5f70<br>\u7b2c8\u56de\u6709\u6a5f\u89e6\u5a92\u30b7\u30f3\u30dd\u30b8\u30a6\u30e0\u3000\u300c\u6709\u6a5f\u5206\u5b50\u89e6\u5a92\u306b\u3088\u308b\u672a\u6765\u578b\u5206\u5b50\u5909\u63db\u300d\u7b2c5\u56de\u516c\u958b\u30b7\u30f3\u30dd\u30b8\u30a6\u30e0\uff0c\u4f9d\u983c\u8b1b\u6f14<br>\u6c96\u7e04\u770c\u5e02\u753a\u6751\u81ea\u6cbb\u4f1a\u9928\u30fb\u81ea\u6cbb\u4f1a\u9928\u30db\u30fc\u30eb\uff0c2015\u5e745\u670810\u65e5<\/li>\n<\/ol>\n\n\n\n<p><\/p>\n\n\n\n<p style=\"font-size:20px\"><strong>2014\u5e74\u5ea6<\/strong><\/p>\n\n\n\n<ol start=\"14\" class=\"wp-block-list\">\n<li>\u300c\u6297\u816b\u760d\u6d3b\u6027\u30a4\u30bd\u30d5\u30e9\u30dc\u30f3\u30fb\u30b0\u30e9\u30b8\u30aa\u30d3\u30a2\u30cb\u30f3 A \u306e\u69cb\u9020\u6d3b\u6027\u76f8\u95a2\u7814\u7a76 (Structure-Activity Relationship Study of Glaziovianin A: An Antitumor Active Isoflavone)\u300d<br>\u7551\u4e2d\u5927\u6210\uff0c\u5869\u7530\u79c0\u4e5f\uff0c\u77e5\u5ff5\u62d3\u5b9f\uff0c\u81fc\u4e95\u5065\u90ce\uff0c\u6728\u8d8a\u82f1\u592b\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c95\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u7406\u5de5\u5b66\u90e8\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0f\u85ac\u5b66\u90e8\uff0c2015\u5e743\u670829\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"13\" class=\"wp-block-list\">\n<li>\u300c\u4e9c\u30ea\u30f3\u9178\u30c8\u30ea\u30a8\u30b9\u30c6\u30eb-\u5c3f\u7d20\u5354\u594f\u89e6\u5a92\u3092\u7528\u3044\u308b 2-\u30b2\u30e9\u30cb\u30eb\u30d5\u30a7\u30ce\u30fc\u30eb\u306e\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u7684\u30d6\u30ed\u30e2\u30dd\u30ea\u30a8\u30f3\u74b0\u5316\u53cd\u5fdc (Phosphite-Urea Cooperative Catalysis for Enantioselective Bromocyclization of 2-Geranylphenols)\u300d<br>\u6fa4\u6751\u6cf0\u5f18\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c95\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u7406\u5de5\u5b66\u90e8\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0f\u85ac\u5b66\u90e8\uff0c2015\u5e743\u670827\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"12\" class=\"wp-block-list\">\n<li>\u300c\u30ad\u30e9\u30eb\u03c0-\u30ab\u30c1\u30aa\u30f3\u89e6\u5a92\u3092\u7528\u3044\u308b\u4e0d\u6589\u74b0\u5316\u4ed8\u52a0\u53cd\u5fdc (Asymmetric Cycloaddition Reactions Induced by Chiral \u03c0-Cation Catalysts)\u300d<br>\u5800\u5c06\u5bdb\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c95\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u7406\u5de5\u5b66\u90e8\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0f\u85ac\u5b66\u90e8\uff0c2015\u5e743\u670826\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"11\" class=\"wp-block-list\">\n<li>\u300c3-\u30d4\u30ed\u30ea\u30f3\u30a2\u30df\u30c9\u306e\u9178\u5316\u7684\u6d3b\u6027\u5316\u3092\u9375\u3068\u3059\u308b\u65b0\u898f\u30de\u30af\u30ed\u30e9\u30af\u30c8 \u30f3\u5316\u6cd5\u306e\u958b\u767a (Development of Macloractonization Based on Oxidative Activation of 3-Pyrroline Amides)\u300d<br>\u5c71\u672c\u5f69\u590f\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c95\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u7406\u5de5\u5b66\u90e8\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0f\u85ac\u5b66\u90e8\uff0c2015\u5e743\u670826\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"10\" class=\"wp-block-list\">\n<li>\u300c\u30cb\u30c8\u30ed\u30a2\u30eb\u30b1\u30f3\u3078\u306e\u03b1-\u30a2\u30df\u30ce\u9178\u30a8\u30b9\u30c6\u30eb\u306e\u30de\u30a4\u30b1\u30eb\u4ed8\u52a0\u3092\u9375 \u53cd\u5fdc\u3068\u3059\u308b\u7f6e\u63db\u30d4\u30da\u30e9\u30b8\u30ce\u30f3\u5408\u6210\u6cd5\u306e\u5fdc\u7528(Application of Substituted Piperazinones Synthesis Based on Michael Addition of \u03b1-Amino Esters to Nitroalkenes)\u300d<br>\u9375\u672c\u7965\u5b50\uff0c\u5de5\u85e4\u5b5d\u5e78\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c95\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u65e5\u672c\u5927\u5b66\u7406\u5de5\u5b66\u90e8\u8239\u6a4b\u30ad\u30e3\u30f3\u30d1\u30b9\uff0f\u85ac\u5b66\u90e8\uff0c2015\u5e743\u670826\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"9\" class=\"wp-block-list\">\n<li>\u300c13-\u30aa\u30ad\u30b7\u30a4\u30f3\u30b2\u30ce\u30fc\u30eb\u306e\u5168\u5408\u6210\u300d<br>\u65e9\u5ddd\u4e00\u90ce<br>\u65e5\u672c\u85ac\u5b66\u4f1a\u7b2c135\u5e74\u4f1a\uff08\u795e\u6238\uff09\uff0c\u30b7\u30f3\u30dd\u30b8\u30a6\u30e0\u300c\u6709\u6a5f\u5408\u6210\u5316\u5b66\u306e\u82e5\u3044\u529b\uff1a\u4eca\uff0c\u3044\u308d\u3093\u306a\u6709\u6a5f\u5316\u5b66\u304c\u9762\u767d\u3044 Young Challengers in Synthetic Organic Chemistry: Diverse Organic Chemistry is Interesting!\u300d\uff0c\u62db\u5f85\u8b1b\u6f14\uff0c\u795e\u6238\uff0c2015\u5e743\u670826\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"8\" class=\"wp-block-list\">\n<li>\"Total synthesis of 13-oxyingenol\"<br>Ichiro Hayakawa<br>\u516c\u76ca\u8ca1\u56e3\u6cd5\u4eba\u30b5\u30f3\u30c8\u30ea\u30fc\u751f\u547d\u79d1\u5b66\u8ca1\u56e3\uff0c\u751f\u6709\u7814\u30b7\u30f3\u30dd\u30b8\u30a6\u30e0\u300c\u5929\u7136\u7269\u6709\u6a5f\u5316\u5b66-\u5206\u5b50\u306e\u529b\u3092\u5f15\u304d\u51fa\u3059-\u300dChemistry of natural products -Power of the molecules-\uff0c\u82f1\u8a9e\u30fb\u62db\u5f85\u8b1b\u6f14\uff0c\u30b5\u30f3\u30c8\u30ea\u30fc\u7814\u7a76\u30bb\u30f3\u30bf\u30fc\uff0c2014\u5e7411\u670817\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"7\" class=\"wp-block-list\">\n<li>\u300c\u30cb\u30c8\u30ed\u30a2\u30eb\u30b1\u30f3\u3078\u306e\u03b1-\u30a2\u30df\u30ce\u9178\u30a8\u30b9\u30c6\u30eb\u306e\u30de\u30a4\u30b1\u30eb\u4ed8\u52a0\u3092\u9375\u53cd\u5fdc\u3068\u3059\u308b\u7f6e\u63db\u30d4\u30da\u30e9\u30b8\u30ce\u30f3\u306e\u65b0\u898f\u5408\u6210\u6cd5\u306e\u958b\u767a\u300d<br>\u5de5\u85e4\u5b5d\u5e78\u3001\u5742\u5009\u5f70<br>\u5ca1\u5c71\u5927\u5b66\u77e5\u6075\u306e\u898b\u672c\u5e022014\uff0c\u53e3\u982d\u8b1b\u6f14\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\u5927\u5b66\u5275\u7acb\uff15\uff10\u5468\u5e74\u8a18\u5ff5\u9928\uff0c2014\u5e7411\u670814\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"6\" class=\"wp-block-list\">\n<li>\u300c\u30cf\u30ed\u30b2\u30f3\u7d50\u5408\u306b\u3088\u308b\u6d3b\u6027\u5316\u3092\u9375\u3068\u3059\u308b\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u7684\u30e8\u30fc\u30c9\u30e9\u30af\u30c8\u30f3\u5316\u53cd\u5fdc\u300d<br>\u5742\u5009\u5f70<br>\u6709\u6a5f\u5206\u5b50\u89e6\u5a92\u306b\u3088\u308b\u672a\u6765\u578b\u5206\u5b50\u5909\u63db\uff0c\u7b2c3\u56de\u6709\u6a5f\u5206\u5b50\u89e6\u5a92\u3000\u82e5\u624b\u30bb\u30df\u30ca\u30fc\uff0c\u7384\u6d77\u30ed\u30a4\u30e4\u30eb\u30db\u30c6\u30eb\uff08\u798f\u5ca1\uff09\uff0c2014\u5e749\u67086\uff0c7\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"5\" class=\"wp-block-list\">\n<li>\u300c\u6297\u816b\u760d\u6027\u30a4\u30bd\u30d5\u30e9\u30dc\u30f3\u30fb\u30b0\u30e9\u30b8\u30aa\u30d3\u30a2\u30cb\u30f3\uff21\u306e\u69cb\u9020\u6d3b\u76f8\u95a2\u7814\u7a76\u300d<br>\u7551\u4e2d\u5927\u6210\uff0c\u65e9\u5ddd\u4e00\u90ce\uff0c\u5742\u5009\u5f70<br>\u7b2c30\u56de\u82e5\u624b\u5316\u5b66\u8005\u306e\u305f\u3081\u306e\u5316\u5b66\u9053\u5834\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u4e0b\u96fb\u30db\u30c6\u30eb\uff08\u5ca1\u5c71\uff09\uff0c2014\u5e748\u670829\uff0c30\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"4\" class=\"wp-block-list\">\n<li>\u300c\u30ad\u30e9\u30eb\u30cb\u30c8\u30ed\u30cd\u30fc\u30c8\u306b\u5bfe\u3059\u308b\u30b8\u30a2\u30b9\u30c6\u30ec\u30aa\u9078\u629e\u7684\u306a\u30d2\u30c9\u30ed\u30ad\u30b7\u30e1\u30c1\u30eb\u5316\u53cd\u5fdc\u306e\u958b\u767a\u3068\u305d\u308c\u3092\u5fdc\u7528\u3057\u305f\u30de\u30f3\u30b6\u30b7\u30b8\u30f3\u5408\u6210\u300d<br>\u4e09\u597d\u590f\u7f8e\uff0c\u5de5\u85e4\u5b5d\u5e78\uff0c\u77f3\u5ddd\u5f70\u5f66\uff0c\u5742\u5009\u5f70<br>\u7b2c30\u56de\u82e5\u624b\u5316\u5b66\u8005\u306e\u305f\u3081\u306e\u5316\u5b66\u9053\u5834\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u4e0b\u96fb\u30db\u30c6\u30eb\uff08\u5ca1\u5c71\uff09\uff0c2014\u5e748\u670829\uff0c30\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"3\" class=\"wp-block-list\">\n<li>\u300c\u6c42\u6838\u89e6\u5a92\u3068\u30eb\u30a4\u30b9\u9178\u306b\u3088\u308b\u5354\u540c\u6d3b\u6027\u5316\u3092\u9375\u3068\u3059\u308b\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u7684\u30e8\u30fc\u30c9\u30e9\u30af\u30c8\u30f3\u5316\u53cd\u5fdc\u300d<br>\u5742\u5009\u5f70<br>\u7b2c30\u56de\u82e5\u624b\u5316\u5b66\u8005\u306e\u305f\u3081\u306e\u5316\u5b66\u9053\u5834\uff0c\u5e2b\u7bc4\u8b1b\u6f14\uff0c\u4e0b\u96fb\u30db\u30c6\u30eb\uff08\u5ca1\u5c71\uff09\uff0c2014\u5e748\u670829\uff0c30\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"2\" class=\"wp-block-list\">\n<li>\u300c\u6c42\u6838\u6027\u6709\u6a5f\u89e6\u5a92\u3092\u7528\u3044\u308b\u9078\u629e\u7684\u30cf\u30ed\u74b0\u5316\u53cd\u5fdc\u300d<br>\u5742\u5009\u5f70<br>\u7b2c49\u56de\u5929\u7136\u7269\u5316\u5b66\u8ac7\u8a71\u4f1a\uff0c\u62db\u5f85\u8b1b\u6f14\uff0c\u305b\u3068\u3046\u3061\u5150\u5cf6\u30db\u30c6\u30eb\uff08\u5ca1\u5c71\uff09\uff0c2014\u5e747\u67082\u301c4\u65e5<\/li>\n<\/ol>\n\n\n\n<ol class=\"wp-block-list\">\n<li>\u300c\u5929\u7136\u7269\u5408\u6210\u3092\u8d77\u70b9\u3068\u3057\u305f\u30b1\u30df\u30ab\u30eb\u30d0\u30a4\u30aa\u30ed\u30b8\u30fc\u30c4\u30fc\u30eb\u306e\u958b\u767a\u7814\u7a76\u300d<br>\u65e9\u5ddd\u4e00\u90ce<br>\u65b0\u5b66\u8853\u9818\u57df\u300c\u5929\u7136\u7269\u30b1\u30df\u30ab\u30eb\u30d0\u30a4\u30aa\u30ed\u30b8\u30fc\u300d\u7b2c5\u56de\u82e5\u624b\u7814\u7a76\u8005\u30ef\u30fc\u30af\u30b7\u30e7\u30c3\u30d7\uff0c\u4f9d\u983c\u8b1b\u6f14\uff0c\u540d\u53e4\u5c4b\u5927\u5b66\u7406\u5b66\u90e8\uff0c2014\u5e745\u670829\u65e5<\/li>\n<\/ol>\n\n\n\n<p><\/p>\n\n\n\n<p style=\"font-size:20px\"><strong>2013\u5e74\u5ea6<\/strong><\/p>\n\n\n\n<p>16.\u300c\u30cb\u30c8\u30ed\u30a2\u30eb\u30b1\u30f3\u3078\u306e\u03b1-\u30a2\u30df\u30ce\u9178\u30a8\u30b9\u30c6\u30eb\u306e\u30de\u30a4\u30b1\u30eb\u4ed8\u52a0\u3092\u9375\u53cd\u5fdc\u3068\u3059\u308b\u7f6e\u63db\u30d4\u30da\u30e9\u30b8\u30ce\u30f3\u306e\u5408\u6210\u300d<br>\u5de5\u85e4\u5b5d\u5e78\uff0c\u78ef\u5c71\u9752\u53f8\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c94\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u540d\u53e4\u5c4b\u5927\u5b66\u6771\u5c71\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2014\u5e743\u670827\u65e5<\/p>\n\n\n\n<p>15.\u300c\u30cb\u30c8\u30ed\u30cd\u30fc\u30c8\u306b\u5bfe\u3059\u308b\u30b8\u30a2\u30b9\u30c6\u30ec\u30aa\u9078\u629e\u7684\u30d2\u30c9\u30ed\u30ad\u30b7\u30e1\u30c1\u30eb\u5316\u3092\u9375\u53cd\u5fdc\u3068\u3059\u308b\u30de\u30f3\u30b6\u30b7\u30b8\u30f3\u306e\u5408\u6210\u7814\u7a76\u300d<br>\u4e09\u597d\u590f\u7f8e\uff0c\u5de5\u85e4\u5b5d\u5e78\uff0c\u77f3\u5ddd\u5f70\u5f66\uff0c\u5742\u5009\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c94\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u540d\u53e4\u5c4b\u5927\u5b66\u6771\u5c71\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2014\u5e743\u670827\u65e5<\/p>\n\n\n\n<p>14.\u300c\u30ad\u30e9\u30eb\u03c0-\u30ab\u30c1\u30aa\u30f3\u89e6\u5a92\u3092\u7528\u3044\u308b\u30a2\u30be\u30e1\u30c1\u30f3\u30a4\u30df\u30f3\u3068\u03b2-\u7f6e\u63db\u30d7\u30ed\u30d4\u30aa\u30ed\u30a4\u30eb\u30d4\u30e9\u30be\u30fc\u30eb\u3068\u306e\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u76841,3-\u53cc\u6975\u5b50\u74b0\u5316\u4ed8\u52a0\u53cd\u5fdc\u300d<br>\u5800\u5c06\u5bdb\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c94\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u540d\u53e4\u5c4b\u5927\u5b66\u6771\u5c71\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2014\u5e743\u670827\u65e5<\/p>\n\n\n\n<p>13.\u300c\u30ad\u30e9\u30ebn-\u30ab\u30c1\u30aa\u30f3\u89e6\u5a92\u306b\u3088\u308b\u30a2\u30ea\u30eb\u30b7\u30e9\u30f3\u3068\u03b1-\u30b1\u30c8\u30a8\u30b9\u30c6\u30eb\u3068\u306e\u30a8\u30ca\u30f3\u30c1\u30aa\u53ca\u3073\u30b8\u30a2\u30b9\u30c6\u30ec\u30aa\u9078\u629e\u7684\u30d8\u30c6\u30edDiels-Alder\u53cd\u5fdc\u306e\u958b\u767a\u300d<br>\u9234\u6728\u8cb4\u5927\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c94\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u540d\u53e4\u5c4b\u5927\u5b66\u6771\u5c71\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2014\u5e743\u670827\u65e5<\/p>\n\n\n\n<p>12.\u300c\u6c42\u6838\u6027\u30ad\u30e9\u30eb\u30ea\u30f3\u9178\u30a8\u30b9\u30c6\u30eb\u89e6\u5a92\u3092\u7528\u3044\u308b\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u7684\u30e8\u30fc\u30c9\u30e9\u30af\u30c8\u30f3\u5316\u53cd\u5fdc\u300d<br>\u4ef2\u8fbb\u79c0\u6587\uff0c\u6fa4\u6751\u6cf0\u5f18\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c94\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u540d\u53e4\u5c4b\u5927\u5b66\u6771\u5c71\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2014\u5e743\u670827\u65e5<\/p>\n\n\n\n<p>11.\u300c\u4e9c\u30ea\u30f3\u9178\u30c8\u30ea\u30a8\u30b9\u30c6\u30eb(III)\u30fc\u5c3f\u7d20\u5354\u594f\u89e6\u5a92\u3092\u7528\u3044\u308b2-\u30b2\u30e9\u30cb\u30eb\u30d5\u30a7\u30ce\u30fc\u30eb\u306e\u9078\u629e\u7684\u30d6\u30ed\u30e2\u30dd\u30ea\u30a8\u30f3\u74b0\u5316\u53cd\u5fdc\u300d<br>\u6fa4\u6751\u6cf0\u5f18\uff0c\u4ef2\u8fbb\u79c0\u6587\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c94\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u540d\u53e4\u5c4b\u5927\u5b66\u6771\u5c71\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2014\u5e743\u670827\u65e5<\/p>\n\n\n\n<p>10.\u300c\u9ad8\u6d3b\u6027\u30ad\u30e9\u30eb\u4e8c\u5869\u57fa\u9178\u89e6\u5a92\u306e\u958b\u767a\uff1a\u5149\u5b66\u6d3b\u6027\u30d4\u30ed\u30ea\u30f3\u9178\u30b8\u30a8\u30b9\u30c6\u30eb\u306e\u5408\u6210\u300d<br>\u5ca1\u672c\u907c\uff0c\u4ef2\u8fbb\u79c0\u6587\uff0c\u5742\u5009\u5f70\uff0c\u6ce2\u591a\u91ce\u5b66\uff0c\u77f3\u539f\u4e00\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c94\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u540d\u53e4\u5c4b\u5927\u5b66\u6771\u5c71\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2014\u5e743\u670827\u65e5<\/p>\n\n\n\n<ol start=\"9\" class=\"wp-block-list\">\n<li>\"Catalytic Asymmetric Cyano-ethoxycarbonylation of Isatns Promoted by Oxyanion Hole Mimetic Lewis Base-Br\u00f8nsted Acid Cooperative Organocatalyst\"<br>Yoshihiro Ogura, Matsujiro Akakura, Akira Sakakura, Kazuaki Ishihara<br>The 3rd Junior International Conference on Cutting-edge Organic Chemistry in Asia, Poster Presentation, Chiba, SEIMEI-NO-MORI, Japan, November 22\u201325, 2013.<\/li>\n<\/ol>\n\n\n\n<ol start=\"8\" class=\"wp-block-list\">\n<li>\"Enantioselective Inverse Electron-Demand Hetero-Diels\u2013Alder Reaction with Allylsilanes\"<br>Akira Sakakura, Yuki Matsumura, Takahiro Suzuki, and Kazuaki Ishihara<br>13th Tateshina Conference on Organic Chemistry, Poster Presentation, Tateshina Forum, November 8\u201310, 2013.<\/li>\n<\/ol>\n\n\n\n<ol start=\"7\" class=\"wp-block-list\">\n<li>\u300c\u6c42\u6838\u6027\u4e9c\u30ea\u30f3\u9178\u30c8\u30ea\u30a8\u30b9\u30c6\u30eb(III)\u89e6\u5a92\u3092\u7528\u3044\u308b\u30dd\u30ea\u30d7\u30ec\u30ce\u30a4\u30c9\u306e\u9078\u629e\u7684\u30d6\u30ed\u30e2\u30dd\u30ea\u30a8\u30f3\u74b0\u5316\u53cd\u5fdc\u300d<br>\u6fa4\u6751\u6cf0\u5f18\u3001\u4ef2\u8fbb\u79c0\u6587\u3001\u5742\u5009\u5f70\u3001\u77f3\u539f\u4e00\u5f70<br>\u7b2c44\u56de\u4e2d\u90e8\u5316\u5b66\u95a2\u4fc2\u5b66\u5354\u4f1a\u652f\u90e8\u9023\u5408\u79cb\u5b63\u5927\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u9759\u5ca1\u5927\u5b66\u6d5c\u677e\u30ad\u30e3\u30f3\u30d1\u30b9\uff0c2013\u5e7411\u67082\u301c3\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"6\" class=\"wp-block-list\">\n<li>\u300c\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u7684\u30e8\u30fc\u30c9\u30e9\u30af\u30c8\u30f3\u5316\u53cd\u5fdc\u306b\u6709\u52b9\u306a\u30ad\u30e9\u30eb\u30ea\u30f3\u6c42\u6838\u89e6\u5a92\u306e\u958b\u767a\u300d<br>\u4ef2\u8fbb\u79c0\u6587\uff0c\u6fa4\u6751\u6cf0\u5f18\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u7b2c30\u56de\u6709\u6a5f\u5408\u6210\u5316\u5b66\u30bb\u30df\u30ca\u30fc\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\uff08\u305b\u3068\u3046\u3061\u5150\u5cf6\u30db\u30c6\u30eb\uff09\uff0c2013\u5e749\u670817\u301c19\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"5\" class=\"wp-block-list\">\n<li>\u300c\u30ad\u30e9\u30ebn-\u30ab\u30c1\u30aa\u30f3\u89e6\u5a92\u306b\u3088\u308b\u30a2\u30ea\u30eb\u30b7\u30e9\u30f3\u306e\u9ad8\u30a8\u30ca\u30f3\u30c1\u30aa\u53ca\u3073\u30b8\u30a2\u30b9\u30c6\u30ec\u30aa\u9078\u629e\u7684\u30d8\u30c6\u30edHetero-Diels\u2013Alder\u53cd\u5fdc\u300d<br>\u9234\u6728\u8cb4\u5927\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u7b2c46\u56de\u6709\u6a5f\u91d1\u5c5e\u82e5\u624b\u306e\u4f1a \u590f\u306e\u5b66\u6821\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5bae\u57ce\uff08\u5bae\u57ce\u8535\u738b\u30ed\u30a4\u30e4\u30eb\u30db\u30c6\u30eb\uff09\uff0c 2013\u5e747\u67088\uff5e10\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"4\" class=\"wp-block-list\">\n<li>\u300c\u751f\u7269\u6d3b\u6027\u30aa\u30ad\u30b7\u30a4\u30f3\u30c9\u30fc\u30eb\u306e\u5408\u6210\u3092\u76ee\u6307\u3057\u305f\u4e0d\u6589\u30b7\u30a2\u30ce\u30a8\u30c8\u30ad\u30b7\u30ab\u30eb\u30dc\u30cb\u30eb\u5316\u53cd\u5fdc\u306e\u958b\u767a\u300d<br>\u5c0f\u5009\u7fa9\u6d69\uff0c\u8d64\u5009\u677e\u6b21\u90ce\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u7b2c48\u56de\u5929\u7136\u7269\u5316\u5b66\u8ac7\u8a71\u4f1a\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u6ecb\u8cc0\uff08\u30a2\u30e4\u30cf\u30ec\u30fc\u30af\u30b5\u30a4\u30c9\u30db\u30c6\u30eb\uff09\uff0c2013\u5e747\u67083\u301c5\u65e5<\/li>\n<\/ol>\n\n\n\n<ol start=\"3\" class=\"wp-block-list\">\n<li>\"Development of Chiral Nucleophilic Phosphite Catalysts for Enantioselective Iodolactonization\"<br>Hidefumi Nakatsuji, Yasuhiro Sawamura, Akira Sakakura, Kazuaki Ishihara<br>Nagoya Symposium 2013, Poster Presentation, Nagoya University, Japan, P-28, May 23, 2013.<\/li>\n<\/ol>\n\n\n\n<ol start=\"2\" class=\"wp-block-list\">\n<li>\"Development of Highly Enantioselective Cyano-Ethoxycarbonylation of Isatin Derivatives\"<br>Yoshihiro Ogura, Matsujiro Akakura, Akira Sakakura, Kazuaki Ishihara<br>Nagoya Symposium 2013, Poster Presentation, Nagoya University, Japan, P-30, May 23, 2013.<\/li>\n<\/ol>\n\n\n\n<ol class=\"wp-block-list\">\n<li>\u300c\u30d0\u30a4\u30aa\u30df\u30e1\u30c6\u30a3\u30c3\u30af\u306a\u30aa\u30ad\u30b5\u30be\u30ea\u30f3\u5408\u6210\u6cd5\u306e\u958b\u767a\u3068\u305d\u306e\u5fdc\u7528\u300d<br>\u5742\u5009\u5f70<br>\u6709\u6a5f\u5408\u6210\u5316\u5b66\u5354\u4f1a\u4e2d\u56fd\u56db\u56fd\u652f\u90e8 \u7b2c68\u56de\u30d1\u30cd\u30eb\u8a0e\u8ad6\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u5ca1\u5c71\uff08\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff09\uff0c2013\u5e745\u670818\u65e5<\/li>\n<\/ol>\n\n\n\n<p><\/p>\n\n\n\n<p style=\"font-size:20px\"><strong>2012\u5e74\u5ea6<\/strong><\/p>\n\n\n\n<p>11.\u300c1,1'-\u30d3\u30ca\u30d5\u30c1\u30eb\u30d4\u30ed\u30ea\u30f3\u9178\u30b8\u30a8\u30b9\u30c6\u30eb\u306e\u5408\u6210\u3068\u30ad\u30e9\u30ebBr\u00f8nsted\u9178\u89e6\u5a92\u3078\u306e\u5c55\u958b (Synthesis of Chiral Binaphthyl Pyrophospate and Development to Chiral Br\u00f8nsted Acid Catalysts)\u300d<br>\u5ca1\u672c\u907c\uff0c\u4ef2\u8fbb\u79c0\u6587\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c93\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6ecb\u8cc0\uff08\u7acb\u547d\u9928\u5927\u5b66\u3073\u308f\u3053\u30fb\u304f\u3055\u3064\u30ad\u30e3\u30f3\u30d1\u30b9\uff09\uff0c3E5-07\uff0c2013\u5e743\u670824\u65e5<\/p>\n\n\n\n<p>10.\u300c\u30a4\u30b5\u30c1\u30f3\u985e\u306e\u9ad8\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u7684\u30b7\u30a2\u30ce\u30a8\u30c8\u30ad\u30b7\u30ab\u30eb\u30dc\u30cb\u30eb\u5316\u53cd\u5fdc\u306e\u958b\u767a (Development of Highly Enantioselective Cyano-Ethoxycarbonylation of Isatin Derivatives)\u300d<br>\u5c0f\u5009\u7fa9\u6d69\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c93\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6ecb\u8cc0\uff08\u7acb\u547d\u9928\u5927\u5b66\u3073\u308f\u3053\u30fb\u304f\u3055\u3064\u30ad\u30e3\u30f3\u30d1\u30b9\uff09\uff0c3E5-06\uff0c2013\u5e743\u670824\u65e5<\/p>\n\n\n\n<p>9.\u300c\u30ad\u30e9\u30eb\u30eb\u30a4\u30b9\u5869\u57fa\u8907\u5408\u578b\u30d6\u30ec\u30f3\u30b9\u30c6\u30c3\u30c9\u9178(LBBA)\u89e6\u5a92\u3092\u7528\u3044\u305f\u4e0d\u6589\u30e9\u30af\u30c8\u30f3\u5316\u306b\u3088\u308b\u30e9\u30bb\u30df\u30ab\u30eb\u30dc\u30f3\u9178\u306e\u901f\u5ea6\u8ad6\u7684\u5149\u5b66\u5206\u5272 (Kinetic Resolution of Racemic Carboxic Acids Catalyzed by Chiral Lewis Base-Assisted Br\u00f8nsted Acid (LBBA) through Asymmetric Lactonization)\u300d<br>\u4f50\u4e45\u9593\u96c5\u5e78\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c93\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6ecb\u8cc0\uff08\u7acb\u547d\u9928\u5927\u5b66\u3073\u308f\u3053\u30fb\u304f\u3055\u3064\u30ad\u30e3\u30f3\u30d1\u30b9\uff09\uff0c2E5-06\uff0c2013\u5e743\u670823\u65e5<\/p>\n\n\n\n<p>8.\u300c\u6c42\u6838\u6027\u4e9c\u30ea\u30f3\u9178\u30a8\u30b9\u30c6\u30eb(III)\u89e6\u5a92\u3092\u7528\u3044\u308b\u30dd\u30ea\u30d7\u30ec\u30ce\u30a4\u30c9\u306e\u9078\u629e\u7684\u30d6\u30ed\u30e2\u30dd\u30ea\u30a8\u30f3\u74b0\u5316\u53cd\u5fdc (Nucleopilic Phosphite(III)-Catalyzed Selective Bromocyclization of Polyprenoids)\u300d<br>\u6fa4\u6751\u6cf0\u5f18\uff0c\u4ef2\u8fbb\u79c0\u6587\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c93\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6ecb\u8cc0\uff08\u7acb\u547d\u9928\u5927\u5b66\u3073\u308f\u3053\u30fb\u304f\u3055\u3064\u30ad\u30e3\u30f3\u30d1\u30b9\uff09\uff0c2E5-05\uff0c2013\u5e743\u670823\u65e5<\/p>\n\n\n\n<p>7.\u300c\u30a8\u30ca\u30f3\u30c1\u30aa\u9078\u629e\u7684\u30e8\u30fc\u30c9\u30e9\u30af\u30c8\u30f3\u5316\u53cd\u5fdc\u306b\u6709\u52b9\u306a\u6c42\u6838\u6027\u30ad\u30e9\u30eb\u4e9c\u30ea\u30f3\u9178\u30a8\u30b9\u30c6\u30eb\u89e6\u5a92\u306e\u958b\u767a (Development of Chiral Nucleophilic Phosphite Catalysts for Enantioselective Iodolactonization)\u300d<br>\u4ef2\u8fbb\u79c0\u6587\uff0c\u6fa4\u6751\u6cf0\u5f18\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c93\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6ecb\u8cc0\uff08\u7acb\u547d\u9928\u5927\u5b66\u3073\u308f\u3053\u30fb\u304f\u3055\u3064\u30ad\u30e3\u30f3\u30d1\u30b9\uff09\uff0c2E5-04\uff0c2013\u5e743\u670823\u65e5<\/p>\n\n\n\n<p>6.\u300c\u30ad\u30e9\u30ebn-\u30ab\u30c1\u30aa\u30f3\u89e6\u5a92\u306b\u3088\u308b\u30a2\u30ea\u30eb\u30b7\u30e9\u30f3\u306e\u9ad8\u30a8\u30ca\u30f3\u30c1\u30aa\u53ca\u3073\u30b8\u30a2\u30b9\u30c6\u30ec\u30aa\u9078\u629e\u7684\u30d8\u30c6\u30edDiels\u2013Alder\u53cd\u5fdc (Highly Enantio- and Diastereoselective Hetero-Diels\u2013Alder Reaction of Allylsilanes Induced by Chiral n-Cation Catalysts)\u300d<br>\u9234\u6728\u8cb4\u5927\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c93\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6ecb\u8cc0\uff08\u7acb\u547d\u9928\u5927\u5b66\u3073\u308f\u3053\u30fb\u304f\u3055\u3064\u30ad\u30e3\u30f3\u30d1\u30b9\uff09\uff0c1E4-33\uff0c2013\u5e743\u670822\u65e5<\/p>\n\n\n\n<p>5.\u300c\u03b1-\u30d2\u30c9\u30ed\u30ad\u30b7\u30ab\u30eb\u30dc\u30f3\u9178\u306e\u30a2\u30df\u30c9\u7e2e\u5408\u306b\u6709\u52b9\u306a\u30dc\u30ed\u30f3\u9178\u89e6\u5a92\u306e\u958b\u767a (Development of Boronic Acid-Catalysts for Amide Condensation of \u03b1-Hydroxycarboxylic Acids)\u300d<br>\u5c71\u4e0b\u8389\u6c99\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>\u65e5\u672c\u5316\u5b66\u4f1a\u7b2c93\u6625\u5b63\u5e74\u4f1a\uff0c\u53e3\u982d\u767a\u8868\uff0c\u6ecb\u8cc0\uff08\u7acb\u547d\u9928\u5927\u5b66\u3073\u308f\u3053\u30fb\u304f\u3055\u3064\u30ad\u30e3\u30f3\u30d1\u30b9\uff09\uff0c1E4-30\uff0c2013\u5e743\u670822\u65e5<\/p>\n\n\n\n<ol start=\"4\" class=\"wp-block-list\">\n<li>\"Template-based de novo design of selective inhibitors of VEGFR-2 kinase\"<br>Takayuki Kudoh<br>The 6th International Symposium for Future Technology Creating Better Human Health and Society, \"Strategies to Establishment Drug Development Systems\" Invited Lecture (Oral Presentation), Graduate School of Natural Science and Technology, Research Building in Okayama University, Japan, February, 7-8, 2013<\/li>\n<\/ol>\n\n\n\n<ol start=\"3\" class=\"wp-block-list\">\n<li>\"Organocatalytic Enantioselective Cyano-Ethoxycarbonylation of Isatins\"<br>Akira Sakakura<br>The 6th International Symposium for Future Technology Creating Better Human Health and Society, \"Strategies to Establishment Drug Development Systems\" Invited Lecture (Oral Presentation), Graduate School of Natural Science and Technology, Research Building in Okayama University, Japan, February, 7-8, 2013<\/li>\n<\/ol>\n\n\n\n<ol start=\"2\" class=\"wp-block-list\">\n<li>\"Enantioselective Organocatalytic Cyanoethoxycarbonylation of Isatin Derivatives\"<br>Akira Sakakura<br>First Japan\u2013USA Organocatalytic Symposium, Invited Lecture (Oral Presentation), Waikiki Prince Hotel, Hawaii, USA, December, 15-18, 2012<\/li>\n<\/ol>\n\n\n\n<ol class=\"wp-block-list\">\n<li>\u300c\u6c42\u6838\u6027\u30ea\u30f3\u9178\u30a8\u30b9\u30c6\u30eb\u89e6\u5a92\u3092\u7528\u3044\u308b\u30dd\u30ea\u30d7\u30ec\u30ce\u30a4\u30c9\u306e\u9078\u629e\u7684\u30dd\u30ea\u30a8\u30f3\u74b0\u5316\u53cd\u5fdc\u300d<br>\u6fa4\u6751\u6cf0\u5f18\uff0c\u4ef2\u8fbb\u79c0\u6587\uff0c\u5742\u5009\u5f70\uff0c\u77f3\u539f\u4e00\u5f70<br>2012 \u30cf\u30ed\u30b2\u30f3\u5229\u7528\u30df\u30cb\u30b7\u30f3\u30dd\u30b8\u30a6\u30e0\uff08\u7b2c5\u56de\u81ed\u7d20\u5316\u5b66\u61c7\u8a71\u4f1a\u5e74\u4f1a\uff09\uff0c\u30dd\u30b9\u30bf\u30fc\u767a\u8868\uff0c\u5ca1\u5c71\uff08\u5ca1\u5c71\u5927\u5b66\u6d25\u5cf6\u30ad\u30e3\u30f3\u30d1\u30b9\uff09\uff0c2012\u5e7411\u670830\u65e5<\/li>\n<\/ol>\n\n\n\n<p><\/p>\n","protected":false},"excerpt":{"rendered":"<p>\u5ca1\u5c71\u5927\u5b66\u5927\u5b66\u9662\u81ea\u7136\u79d1\u5b66\u7814\u7a76\u79d1\u3000\u751f\u7269\u6709\u6a5f\u5316\u5b66\u7814\u7a76\u5ba4\uff08\u5742\u5009\u7814\u7a76\u5ba4\uff09\u306eHP\u3067\u3059\u3002\u5f53\u7814\u7a76\u5ba4\u3067\u306f\u3001\u5929\u7136\u6709\u6a5f\u5316\u5408\u7269\u306b\u5b66\u3073\u306a\u304c\u3089\u3001\u7acb\u4f53\u9078\u629e\u7684\u306a\u53cd\u5fdc\u3092\u53ef\u80fd\u3068\u3059\u308b\u30eb\u30a4\u30b9\u9178\u89e6\u5a92\u3084\u6709\u6a5f\u5206\u5b50\u89e6\u5a92\u306e\u958b\u767a\u30db\u30a6\u7d20\u306e\u7279\u6027\u3092\u751f\u304b\u3057\u305f\u53cd\u5fdc\u958b\u767a\u751f\u7269\u6d3b\u6027\u5206\u5b50\u306e\u5408\u6210\u306a\u3069\u306b\u53d6\u308a\u7d44\u3093\u3067\u3044\u307e\u3059\uff01\uff01<\/p>\n","protected":false},"author":1,"featured_media":0,"parent":0,"menu_order":0,"comment_status":"closed","ping_status":"closed","template":"","meta":{"vkexunit_cta_each_option":"","footnotes":""},"class_list":["post-203","page","type-page","status-publish","hentry"],"_links":{"self":[{"href":"http:\/\/achem.okayama-u.ac.jp\/bioorgchem\/wp-json\/wp\/v2\/pages\/203","targetHints":{"allow":["GET"]}}],"collection":[{"href":"http:\/\/achem.okayama-u.ac.jp\/bioorgchem\/wp-json\/wp\/v2\/pages"}],"about":[{"href":"http:\/\/achem.okayama-u.ac.jp\/bioorgchem\/wp-json\/wp\/v2\/types\/page"}],"author":[{"embeddable":true,"href":"http:\/\/achem.okayama-u.ac.jp\/bioorgchem\/wp-json\/wp\/v2\/users\/1"}],"replies":[{"embeddable":true,"href":"http:\/\/achem.okayama-u.ac.jp\/bioorgchem\/wp-json\/wp\/v2\/comments?post=203"}],"version-history":[{"count":15,"href":"http:\/\/achem.okayama-u.ac.jp\/bioorgchem\/wp-json\/wp\/v2\/pages\/203\/revisions"}],"predecessor-version":[{"id":512,"href":"http:\/\/achem.okayama-u.ac.jp\/bioorgchem\/wp-json\/wp\/v2\/pages\/203\/revisions\/512"}],"wp:attachment":[{"href":"http:\/\/achem.okayama-u.ac.jp\/bioorgchem\/wp-json\/wp\/v2\/media?parent=203"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}