2021年11月

2018年度
Thioureas as Highly Active Catalysts for Biomimetic Bromocyclization of Geranyl Derivatives

Miyuki Terazaki, Kei-ichi Shiomoto, Haruki Mizoguchi, Akira Sakakura* Org. Lett.2019, 21 (7), 2 […]

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2018年度
Catalytic Enantioselective Hosomi–Sakurai Reaction of α-Ketoesters Promoted by Chiral Copper(II) Complexes

Yutaro Niwa, Mayu Miyake, Ichiro Hayakawa, Akira Sakakura* Chem. Commun.2019, 55 (27), 3923–392 […]

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2018年度
Chiral Pyrophosphoric Acid Catalysts for the para-Selective and Eanantioselective Aza-Friedel–Crafts Reaction of Phenols

Haruka Okamoto, Kohei Toh, Takuya Mochizuki, Hidefumi Nakatsuji, Akira Sakakura,* Manabu Hatano,* Kazuaki Ishi […]

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2018年度
Enantioselective aza-Friedel–Crafts reaction of furan with α-ketimino esters induced by a conjugated double hydrogen bond network of chiral bis(phosphoric acid) catalysts

Manabu Hatano,  Haruka Okamoto,  Taro Kawakami,  Kohei Toh,  Hidefumi Nakatsuji,  Aki […]

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2017年度
Regioselective DMAD-insertion Reaction of Silyl Dienol Ether of γ-Pyrone under Catalyst- and Heating-Free Conditions

Ichiro Hayakawa,* Yuji Yamanaka, Koichi Mitsudo, Hiromi Ota, Akira Sakakura* Heterocycles2017, 94&nb […]

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2017年度
Diastereodivergent Henry Reaction for the Stereoselective Construction of Nitrogen-Containing Tetrasubstituted Carbons: Application to Total Synthesis of Manzacidins A and C

Takayuki Kudoh, Yuya Araki, Natsumi Miyoshi, Mizuho Tanioka, and Akira Sakakura* Asian J. Org. Chem.2017, […]

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2017年度
Heat Versus Basic Conditions: Intramolecular Dehydro-Diels–Alder Reaction of 1-Indolyl-1,6-heptadiynes for the Selective Synthesis of Substituted Carbazoles

Takayuki Kudoh, Syo Fujisawa, Megumi Kitamura, Akira Sakakura* Synlett2017, 28 (16), 2189–2193. […]

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2017年度
Reinvestigation of the Biomimetic Cyclization of 3,5-Diketoesters: Application to the Total Synthesis of Cyercene A, an α-Methoxy-γ-Pyrone-Containing Polypropionate

Kai Onda, Ichiro Hayakawa, Akira Sakakura*Synlett2017, 28 (13), 1596–1600.  (Published online: […]

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2017年度
Copper(II) Triflimide

Akira Sakakura, Kazuaki IshiharaIn e-EROS (Encyclopedia of Reagents for Organic Synthesis); Wiley, 2 […]

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2016年度
Discovery of O6-benzyl glaziovianin A, a potent cytotoxic substance and a potent inhibitor of α,β-tubulin polymerization

Ichiro Hayakawa,* Shuya Shioda, Takumi Chinen, Taisei Hatanaka, Haruna Ebisu, Akira Sakakura, Takeo Usui,* Hid […]

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