Enantioselective construction of β-hydroxy-α,α-disubstituted α-amino acid derivatives via direct aldol reaction of α-imino esters
Yuya Araki, Masato Hanada, Yoshiko Iguchi, Haruki Mizoguchi, Akira Sakakura*Tetrahedron, in Press DOI: 10.1016 […]
Toward the Synthesis of Paspaline-Type Indole-Terpenes: Stereoselective Construction of Core Scaffold with Contiguous Asymmetric Quaternary Carbon Centers
Ichiro Hayakawa*, Naochika Matsumaru, and Akira Sakakura* J. Org. Chem.2021, ASAP (Published online: July […]
Strain-Release Difunctionalization of C–C σ- and π-bonds of an Organoboron Ate-Complex through 1,2-Metallate Rearrangement
Haruki Mizoguchi,* Akira Sakakura* Chem. Lett.2021, 50 (4), 792–799. (Published online: January […]
Synthesis of functionalized cyclopropylboronic esters based on a 1,2-metallate rearrangement of cyclopropenylboronate
Haruki Mizoguchi,* Masaya Seriua, Akira Sakakura* Chem. Commun.2020, 56 (99), 15545–15548. (Pub […]
Kinetic Resolution of α-Nitrolactones by Catalytic Asymmetric Hydrolysis or Ester–Amide Exchange Reaction
Ryota Nakao, Yudai Fujii, Ichiro Hayakawa, Haruki Mizoguchi, Akira Sakakura* Synlett2020, 31 (2 […]
Enantioselective Diels–Alder Reaction of 3-Nitrocoumarins Promoted by Chiral Organoammonium Salt Catalysts
Yudai Fujii, Ryota Nakao, Saki Sugihara, Keita Fujita, Yuya Araki, Takayuki Kudoh, Ichiro Hayakawa, Haruki Miz […]
Structure Optimization of Gatastatin for the Development of γ-Tubulin-Specific Inhibitor
Kana Shintani, Haruna Ebisu, Minagi Mukaiyama, Taisei Hatanaka, Takumi Chinen, Daisuke Takao, Yoko Nagumo, Aki […]
Formal Total Synthesis of Manzacidin B via Sequential Diastereodivergent Henry Reaction
Yuya Araki, Natsumi Miyoshi, Kazuki Morimoto, Takayuki Kudoh, Haruki Mizoguchi, Akira Sakakura* J. Org. C […]
Toward the Synthesis of SB-203207: Construction of Four Contiguous Nitrogen-Containing Stereogenic Centers
Ichiro Hayakawa,* Anna Nagayasu, Akira Sakakura*J. Org. Chem.2019, 84 (23), 15614–15623. (Published […]